SCHEMBL9539833

SCHEMBL9539833

COc1ccc(CN2CCCCC2c2ccccc2)cc1

nearest known ligand 0.58

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.58
OPRK1 P41145 3/20 0.57
OPRM1 P35372 2/20 0.57
KDM4E B2RXH2 1/20 0.57
ALDH1A1 P00352 1/20 0.57
HRH2 P25021 1/20 0.55
HCRTR1 O43613 1/20 0.54
GAA P10253 1/20 0.50
KMT2A Q03164 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24365232 0.85 KDM4E (0.56) OPRK1OPRM1KDM4EALDH1A1GAA
SCHEMBL11488897 0.85 KDM4E (0.56) OPRK1OPRM1KDM4EALDH1A1GAA
SCHEMBL23747732 0.82 OPRK1 (0.52) SIGMAR1OPRK1OPRM1KDM4EALDH1A1
SCHEMBL8543954 0.82 KDM4E (0.64) SIGMAR1OPRK1OPRM1KDM4EALDH1A1
SCHEMBL7189631 0.81 OPRK1 (0.55) OPRK1OPRM1KDM4EALDH1A1KMT2A
SCHEMBL2172790 0.81 CHRNB2 (0.53) OPRK1OPRM1KDM4EALDH1A1GAA
SCHEMBL22201130 0.81 CHRNB2 (0.53) OPRK1OPRM1KDM4EALDH1A1GAA
SCHEMBL11707128 0.80 SIGMAR1 (0.51) SIGMAR1OPRK1OPRM1HRH2
SCHEMBL23747503 0.80 NPC1 (0.60) OPRK1OPRM1KDM4EALDH1A1KMT2A
SCHEMBL23747504 0.80 NPC1 (0.60) OPRK1OPRM1KDM4EALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993004040-A1 AZACYCLIC COMPOUNDS, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM MERCK SHARP & DOHME LIMITED (GB) 1993-03-04 WO claimed