SCHEMBL9539840

SCHEMBL9539840

CCCCC(=O)Nc1ccc(C(F)(F)F)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.65
ALDH1A1 P00352 3/20 0.65
MAPT P10636 1/20 0.65
MEN1 O00255 3/20 0.60
KMT2A Q03164 3/20 0.60
HTT P42858 2/20 0.60
LMNA P02545 1/20 0.60
RORC P51449 3/20 0.58
CA12 O43570 1/20 0.57
CA1 P00915 1/20 0.57
CA2 P00918 1/20 0.57
CA9 Q16790 1/20 0.57
EPHX2 P34913 1/20 0.56
KCNQ3 O43525 1/20 0.55
KCNQ2 O43526 1/20 0.55
KCNQ4 P56696 1/20 0.55
KCNQ5 Q9NR82 1/20 0.55
CYP2D6 P10635 2/20 0.54
CYP2C19 P33261 2/20 0.54
CYP3A4 P08684 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9842932 0.90 TP53 (0.66) SMN1; SMN2ALDH1A1MAPTMEN1KMT2A
SCHEMBL23054850 0.88 EPHX2 (0.61) EPHX2L3MBTL1
SCHEMBL8171576 0.86 RORC (0.59) SMN1; SMN2ALDH1A1MAPTMEN1KMT2A
SCHEMBL7368975 0.86 RORC (0.56) SMN1; SMN2ALDH1A1MAPTMEN1KMT2A
SCHEMBL24590188 0.85 ALDH1A1 (0.59) SMN1; SMN2ALDH1A1MEN1KMT2ACA12
SCHEMBL19370084 0.85 CNR1 (0.73) ALDH1A1MAPTMEN1KMT2ACYP2C19
SCHEMBL16229451 0.85 SIRT1 (0.64) SMN1; SMN2ALDH1A1MAPT
SCHEMBL15480429 0.84 HDAC1 (0.68) ALDH1A1MEN1KMT2AHTTLMNA
SCHEMBL22298749 0.84 KCNQ3 (0.59) SMN1; SMN2ALDH1A1MAPTMEN1KMT2A
SCHEMBL5541646 0.84 EPHX2 (0.56) SMN1; SMN2ALDH1A1MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114751874-B 1-Benzyl-4-ethylpiperazine derivatives as TRPV4-KCa2.3 coupling promoters and uses thereof 江南大学 2025-01-24 CN disclosed
CN-114751874-A 1-benzyl-4-ethylpiperazine derivatives as TRPV4-KCa2.3 coupling promoting agents and application thereof 江南大学 2022-07-15 CN disclosed
WO-1993013766-A1 TREATMENT OF INVOLUNTARY MOVEMENTS WITH 5HT1A RECEPTOR AGONISTS MERRELL DOW PHARMACEUTICALS INC. (US) 1993-07-22 WO disclosed
EP-0440503-A1 4-Isoxazolecarboxamide derivatives SYNTEX (U.S.A.) INC. (US) 1991-08-07 EP disclosed