SCHEMBL9539867

SCHEMBL9539867

O=C(O)c1c(Cc2ccc(Br)cc2)[nH]c(=O)c2ccccc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.46
MAOB P27338 1/20 0.43
KDM4E B2RXH2 3/20 0.41
TDP1 Q9NUW8 1/20 0.41
PARP1 P09874 3/20 0.40
TNKS O95271 1/20 0.40
CYP1A1 P04798 1/20 0.40
CYP1B1 Q16678 1/20 0.40
TNKS2 Q9H2K2 1/20 0.40
VKORC1 Q9BQB6 1/20 0.39
PDE3B Q13370 1/20 0.39
PDE3A Q14432 1/20 0.39
AKR1C3 P42330 1/20 0.39
KMT2A Q03164 3/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
ALDH1A1 P00352 2/20 0.37
MEN1 O00255 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5510275 0.73 KDM4E (0.56) ALOX5KDM4ETDP1KMT2AALDH1A1
SCHEMBL9541424 0.70 KDM4E (0.42) KDM4ETDP1PARP1TNKSTNKS2
SCHEMBL31716910 0.69 KMT2A (0.80) MAOBKDM4EPARP1TNKSCYP1A1
SCHEMBL7696486 0.69 ALDH1A1 (0.54) KDM4ETDP1KMT2AALDH1A1MEN1
SCHEMBL9541047 0.68 LOXL2 (0.57) MAOBKDM4EPARP1TNKSCYP1A1
SCHEMBL31716561 0.68 LOXL2 (0.57) MAOBKDM4EPARP1TNKSCYP1A1
SCHEMBL9540970 0.68 GPR17 (0.52) PDE3BPDE3A
SCHEMBL9542605 0.68 ALOX5 (0.42) ALOX5MAOBKDM4EPARP1TNKS
SCHEMBL7823681 0.67 KDM4E (0.51) KDM4ETDP1PARP1TNKSTNKS2
SCHEMBL6605700 0.66 MEN1 (0.47) MAOBKDM4ETDP1PARP1VKORC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993014086-A1 SUBSTITUTED 1-ISOQUINOLONE DERIVATIVES AS ANGIOTENSIN II ANTAGONISTS SYNTEX (U.S.A.) INC. (US) 1993-07-22 WO disclosed