SCHEMBL9540210

SCHEMBL9540210

Clc1ccc(C=P(c2ccccc2)(c2ccccc2)c2ccccc2)c(Cl)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.47
CYP1A2 P05177 1/20 0.39
CYP2C19 P33261 1/20 0.39
MAPT P10636 5/20 0.39
LMNA P02545 4/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
HTT P42858 3/20 0.39
HPGD P15428 3/20 0.39
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 2/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
ALPL P05186 1/20 0.39
GLA P06280 1/20 0.39
GAA P10253 1/20 0.39
ALPG P10696 1/20 0.39
PKM P14618 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
GRIN2D O15399 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9538666 0.78 NPBWR1 (0.39) MAPTLMNAMEN1KMT2AHTT
SCHEMBL9541503 0.72 TSHR (0.42) CYP1A2MAPTLMNAHSD17B10
SCHEMBL3295740 0.71 TDP1 (0.52) TDP1CYP1A2CYP2C19MAPTLMNA
SCHEMBL722335 0.69 NPC1 (0.51) TDP1MAPTLMNAMEN1KMT2A
SCHEMBL722334 0.69 NPC1 (0.51) TDP1MAPTLMNAMEN1KMT2A
SCHEMBL27686167 0.68 TDP1 (0.54) TDP1CYP1A2CYP2C19MAPTLMNA
SCHEMBL2097650 0.68 TDP1 (0.65) TDP1MAPTALDH1A1KDM4ENPC1
SCHEMBL9538195 0.68 ALDH1A1 (0.45) MAPTLMNAMEN1KMT2AALDH1A1
Styrene SCHEMBL9066030 0.67 ALDH1A1 (0.52) TDP1CYP1A2CYP2C19MAPTLMNA
SCHEMBL10743224 0.67 CYP1A2 (0.58) TDP1CYP1A2CYP2C19MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0311955-B1 BICYCLIC PEROXIDE F. HOFFMANN-LA ROCHE AG (CH) 1993-04-21 EP disclosed
US-5134240-A Malaria therapy HOFFMANN-LAROCHE, INC. (US) 1992-07-28 US disclosed
US-4977184-A Bicyclic peroxides compositions for and treatment of malaria therewith HOFFMANN-LA ROCHE INC. (US) 1990-12-11 US disclosed
EP-0311955-A2 Bicyclic peroxide F. HOFFMANN-LA ROCHE AG (CH) 1989-04-19 EP disclosed