SCHEMBL9541503

SCHEMBL9541503

Clc1ccc(C=P(c2ccccc2)(c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.42
CYP1A2 P05177 1/20 0.41
G6PC1 P35575 1/20 0.41
MAPT P10636 1/20 0.40
HSD17B10 Q99714 1/20 0.39
MAOB P27338 2/20 0.39
G6PD P11413 1/20 0.37
NFE2L2 Q16236 1/20 0.37
EGFR P00533 1/20 0.36
MMP1 P03956 1/20 0.36
MMP2 P08253 1/20 0.36
MMP9 P14780 1/20 0.36
PTGS2 P35354 1/20 0.36
AHR P35869 1/20 0.35
FBP1 P09467 1/20 0.35
IDO1 P14902 1/20 0.35
TDO2 P48775 1/20 0.35
CYP1B1 Q16678 1/20 0.35
SIRT1 Q96EB6 1/20 0.35
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1132385 0.84 ALDH1A1 (0.39) TSHRCYP1A2MAPTMAOBNFE2L2
SCHEMBL9539397 0.80 ALDH1A1 (0.41) CYP1A2MAPTHSD17B10SIRT1LMNA
SCHEMBL14269409 0.78 ALDH1A1 (0.42) MAPTMAOBG6PDCYP1B1LMNA
SCHEMBL9538596 0.78 LMNA (0.42) TSHRMAPTNFE2L2EGFRMMP1
SCHEMBL9541494 0.78 NFE2L2 (0.52) TSHRMAPTNFE2L2EGFRMMP1
SCHEMBL24193844 0.78 ESR1 (0.50) G6PC1MAPTNFE2L2MMP1MMP2
SCHEMBL9538195 0.78 ALDH1A1 (0.45) TSHRG6PC1MAPTAHRIDO1
SCHEMBL14423637 0.75 LTA4H (0.48) TSHRMMP2LMNA
Benzaldehyde SCHEMBL6051056 0.74 ALDH1A1 (0.61) TSHRHSD17B10MAOBFBP1LMNA
SCHEMBL9538770 0.74 TRPV1 (0.41) TSHRCYP1A2MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0311955-B1 BICYCLIC PEROXIDE F. HOFFMANN-LA ROCHE AG (CH) 1993-04-21 EP disclosed
US-5134240-A Malaria therapy HOFFMANN-LAROCHE, INC. (US) 1992-07-28 US disclosed
US-4977184-A Bicyclic peroxides compositions for and treatment of malaria therewith HOFFMANN-LA ROCHE INC. (US) 1990-12-11 US disclosed
EP-0311955-A2 Bicyclic peroxide F. HOFFMANN-LA ROCHE AG (CH) 1989-04-19 EP disclosed
US-4065620-A ANTIBIOTICS ELI LILLY AND COMPANY (US) 1977-12-27 US disclosed