SCHEMBL9540305

SCHEMBL9540305

CCCCCCCCC(C)CC(Cc1csc2ccccc12)(OC(N)=O)C(=O)NC(CO)Cc1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSL P07711 1/20 0.35
CTSS P25774 1/20 0.35
CTSK P43235 1/20 0.35
CYP3A4 P08684 1/20 0.35
MAPK1 P28482 1/20 0.35
TACR1 P25103 1/20 0.34
DYRK1A Q13627 1/20 0.33
DYRK1B Q9Y463 1/20 0.33
PIN1 Q13526 1/20 0.33
CSNK1E P49674 1/20 0.33
OPRM1 P35372 2/20 0.33
OPRD1 P41143 2/20 0.33
OPRK1 P41145 2/20 0.33
CTSG P08311 2/20 0.32
CMA1 P23946 2/20 0.32
MME P08473 1/20 0.32
MMP1 P03956 1/20 0.32
MMP2 P08253 1/20 0.32
MMP3 P08254 1/20 0.32
MMP7 P09237 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9540187 0.85 PARP1 (0.35) CTSLCTSKCYP3A4MAPK1CSNK1E
SCHEMBL9538885 0.78 GABRA1 (0.40) CYP3A4
SCHEMBL9540034 0.78 CYP3A4 (0.36) CTSLCTSSCTSKCYP3A4MAPK1
SCHEMBL9539180 0.64 MMP8 (0.44) CTSLCTSSCTSKCYP3A4OPRK1
SCHEMBL4899214 0.64 CTSS (0.63) CTSLCTSSCTSKCYP3A4TACR1
SCHEMBL4900597 0.64 CTSS (0.63) CTSLCTSSCTSKCYP3A4TACR1
SCHEMBL6855159 0.64 CTSS (0.63) CTSLCTSSCTSKCYP3A4TACR1
SCHEMBL27133307 0.64 CYP2A6 (0.53) CTSLCTSSCTSKTACR1OPRM1
SCHEMBL27032777 0.64 CYP2A6 (0.53) CTSLCTSSCTSKTACR1OPRM1
SCHEMBL6888466 0.63 USP2 (0.47) CYP3A4MAPK1TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993003721-A1 CHOLECYSTOKININ ANTAGONISTS USEFUL FOR TREATING DEPRESSION WARNER-LAMBERT COMPANY (US) 1993-03-04 WO claimed