SCHEMBL9540187

SCHEMBL9540187

CCCCCCCCC(C)CC(Cc1ccnc2ccccc12)(OC(N)=O)C(=O)NC(CO)Cc1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.35
PARP3 Q9Y6F1 1/20 0.35
CYP3A4 P08684 1/20 0.35
MAPK1 P28482 1/20 0.35
ITGB1 P05556 1/20 0.34
ITGA4 P13612 1/20 0.34
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33
CCR1 P32246 1/20 0.33
CSNK1E P49674 1/20 0.33
TACR3 P29371 1/20 0.33
TLR8 Q9NR97 2/20 0.33
CTSK P43235 2/20 0.33
TLR7 Q9NYK1 1/20 0.33
CTSL P07711 1/20 0.33
CTSB P07858 1/20 0.33
CTSH P09668 1/20 0.33
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
MAPT P10636 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9540305 0.85 CTSL (0.35) CYP3A4MAPK1CSNK1ECTSKCTSL
SCHEMBL9538885 0.81 GABRA1 (0.40) CYP3A4KDM4EMEN1MAPTKMT2A
SCHEMBL9540182 0.78 KDM4E (0.41) ITGB1ITGA4TACR3CTSKCTSL
SCHEMBL9698405 0.72 KDM4E (0.45) PARP1PARP3CYP3A4MAPK1CCR1
SCHEMBL9699633 0.69 MAPK1 (0.47) PARP1PARP3CYP3A4MAPK1CCR1
SCHEMBL9537553 0.65 MAPK1 (0.43) CYP3A4MAPK1MAPTKMT2A
SCHEMBL7665154 0.64 CCKBR (0.35) PARP1PARP3CYP3A4MAPK1CCR1
SCHEMBL9538450 0.63 KDM4E (0.42) CYP3A4MAPK1TACR3CTSKCTSL
SCHEMBL6888466 0.63 USP2 (0.47) CYP3A4MAPK1KDM4EMEN1MAPT
SCHEMBL3403504 0.62 CSNK1E (0.54) CNR2CSNK1E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993003721-A1 CHOLECYSTOKININ ANTAGONISTS USEFUL FOR TREATING DEPRESSION WARNER-LAMBERT COMPANY (US) 1993-03-04 WO disclosed