SCHEMBL9541244

SCHEMBL9541244

CC1=C2CC[C@@H]3[C@H](CC[C@@]4(C)[C@H]3C=C[C@]4(C)O)[C@H]2CC/C1=N\O

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 3/20 0.35
PDK2 Q15119 3/20 0.35
PDK3 Q15120 3/20 0.35
PDK4 Q16654 3/20 0.35
PGR P06401 2/20 0.31
AR P10275 2/20 0.31
LMNA P02545 1/20 0.31
ESR1 P03372 1/20 0.31
SLC6A4 P31645 1/20 0.31
OPRM1 P35372 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9542392 0.84 PGR (0.41) PGRARLMNAESR1SLC6A4
SCHEMBL9541221 0.84
SCHEMBL9541223 0.78 PDK1 (0.43) PDK1PDK2PDK3PDK4PGR
SCHEMBL9542422 0.74 CYP3A4 (0.39) PGRARLMNAESR1
SCHEMBL9541199 0.71 PGR (0.58) PGRARLMNAESR1SLC6A4
SCHEMBL9128149 0.69 CYP3A4 (0.36) PGRARLMNAESR1
SCHEMBL9128153 0.69 CYP3A4 (0.36) PGRARLMNAESR1
SCHEMBL9541966 0.65 PDK1 (0.43) PDK1PDK2PDK3PDK4PGR
SCHEMBL9124545 0.65 SHBG (0.43) PGRARLMNAESR1
SCHEMBL9124551 0.65 SHBG (0.43) PGRARLMNAESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993013122-A1 3-METHYLSULPHONYLHYDRAZONO AND 3-OXYIMINO STEROIDS, A METHOD OF PREPARING THEM, PHARMACEUTICAL PREPARATIONS CONTAINING THEM AND THEIR USE IN THE PREPARATION OF DRUGS SCHERING AKTIENGESELLSCHAFT (DE) 1993-07-08 WO claimed
WO-1993013122-A1 3-METHYLSULPHONYLHYDRAZONO AND 3-OXYIMINO STEROIDS, A METHOD OF PREPARING THEM, PHARMACEUTICAL PREPARATIONS CONTAINING THEM AND THEIR USE IN THE PREPARATION OF DRUGS SCHERING AKTIENGESELLSCHAFT (DE) 1993-07-08 WO disclosed