SCHEMBL9541340

SCHEMBL9541340

CC=Cn1c(Cc2ccc(Br)cc2)c(C(=O)O)c2ccccc2c1=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 1/20 0.37
PDE3A Q14432 1/20 0.37
VKORC1 Q9BQB6 1/20 0.34
FPR1 P21462 1/20 0.34
FPR2 P25090 1/20 0.34
GPR52 Q9Y2T5 1/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
KDM4E B2RXH2 1/20 0.34
RECQL P46063 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
AKR1C3 P42330 1/20 0.33
TSHR P16473 1/20 0.33
ERCC5 P28715 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9542658 0.79 MAPT (0.36) ALDH1A1NPSR1KMT2AKDM4ETSHR
SCHEMBL9542617 0.76 TDP1 (0.50) MEN1KMT2AKDM4ETDP1L3MBTL1
SCHEMBL9541379 0.73 GPR17 (0.41) PDE3BPDE3AMEN1KMT2A
SCHEMBL9539844 0.72 PDE3B (0.37) PDE3BPDE3AVKORC1FPR1MEN1
SCHEMBL9542653 0.70 KDM4E (0.33) ALDH1A1NPSR1MEN1KMT2AKDM4E
SCHEMBL9539867 0.66 ALOX5 (0.46) PDE3BPDE3AVKORC1ALDH1A1MEN1
SCHEMBL2676347 0.64 MAPK1 (0.51) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL2676056 0.62 ALDH1A1 (0.47) ALDH1A1NPSR1MEN1KMT2AKDM4E
SCHEMBL2676368 0.61 MAPK1 (0.51) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL2677820 0.61 MAPK1 (0.47) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993014086-A1 SUBSTITUTED 1-ISOQUINOLONE DERIVATIVES AS ANGIOTENSIN II ANTAGONISTS SYNTEX (U.S.A.) INC. (US) 1993-07-22 WO disclosed