SCHEMBL9541716

SCHEMBL9541716

CCC(=Cc1cnc2nc(N)nc(N)c2n1)c1ccc(C(=O)OC)cc1

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DHFR P00374 13/20 0.43
ROCK1 Q13464 1/20 0.41
NPC1 O15118 1/20 0.38
TP53 P04637 1/20 0.38
GLA P06280 1/20 0.38
MAPK1 P28482 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9543422 1.00 DHFR (0.43) DHFRROCK1NPC1TP53GLA
SCHEMBL9541711 0.81 DHFR (0.41) DHFR
SCHEMBL9541721 0.81 DHFR (0.41) DHFR
SCHEMBL9544503 0.80 DHFR (0.40) DHFRNPC1TP53GLAMAPK1
SCHEMBL9541999 0.73 DHFR (0.66) DHFR
SCHEMBL9542041 0.72 DHFR (0.52) DHFR
SCHEMBL9542054 0.72 DHFR (0.47) DHFR
SCHEMBL9547681 0.68 DHFR (0.45) DHFR
SCHEMBL3769952 0.67 NOS1 (0.47) DHFRNPC1TP53GLAMAPK1
SCHEMBL9314999 0.67 DHFR (0.47) DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993013102-A1 DEAZAAMINOPTERINS SOUTHERN RESEARCH INSTITUTE (US) 1993-07-08 WO claimed
WO-1993013102-A1 DEAZAAMINOPTERINS SOUTHERN RESEARCH INSTITUTE (US) 1993-07-08 WO disclosed
WO-1993013102-A1 DEAZAAMINOPTERINS SOUTHERN RESEARCH INSTITUTE (US) 1993-07-08 WO disclosed
US-5077404-A Cyclized 5,10-dideazaaminopterin compounds SRI INTERNATIONAL 1991-12-31 US disclosed
US-5077404-A Cyclized 5,10-dideazaaminopterin compounds SRI INTERNATIONAL 1991-12-31 US disclosed