SCHEMBL9543615

SCHEMBL9543615

CC(C)(C)OC(=O)N(C(=O)[C@@H]1C[C@H](Oc2ccccn2)CCN1)C(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.42
EPHX2 P34913 1/20 0.35
PIM2 Q9P1W9 3/20 0.35
PIM1 P11309 2/20 0.35
NAAA Q02083 1/20 0.35
KDM5A P29375 1/20 0.35
GPR119 Q8TDV5 2/20 0.34
HCRTR1 O43613 2/20 0.34
HCRTR2 O43614 2/20 0.34
AVPR1A P37288 4/20 0.33
SCN9A Q15858 1/20 0.33
FFAR1 O14842 2/20 0.33
IP6K1 Q92551 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9543647 0.74 GRIK1 (0.33) GPR119
SCHEMBL9543675 0.72 ELOVL6 (0.33)
SCHEMBL15625371 0.70 EPHX2 (0.41) HRH3EPHX2NAAAKDM5AGPR119
SCHEMBL7420310 0.69 SCN4A (0.43) SCN9A
SCHEMBL12094627 0.68 GPR119 (0.61) NAAAGPR119
SCHEMBL29749275 0.67 GPR119 (0.62) EPHX2KDM5AGPR119
SCHEMBL1087898 0.67 GPR119 (0.62) EPHX2KDM5AGPR119
Acetic Acid SCHEMBL4325103 0.67 HRH1 (0.49) EPHX2NAAAKDM5AHCRTR1HCRTR2
SCHEMBL6344507 0.67 EPHX2 (0.44) EPHX2KDM5AGPR119
SCHEMBL3001240 0.67 GPR119 (0.52) EPHX2KDM5AGPR119HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993018003-A1 SUBSTITUED PIPECOLINIC ACID DERIVATIVES AS HIV PROTEASE INHIBITORS BIO-MEGA/BOEHRINGER INGELHEIM RESEARCH INC. (CA) 1993-09-16 WO disclosed