SCHEMBL9543635

SCHEMBL9543635

COC(=O)CCc1ccc(CCl)c(Cl)c1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PYGL P06737 1/20 0.44
TSHR P16473 1/20 0.42
PTPN1 P18031 2/20 0.41
KMT2A Q03164 1/20 0.41
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
MAPT P10636 1/20 0.40
IDO1 P14902 1/20 0.40
SIRT2 Q8IXJ6 1/20 0.40
CDK8 P49336 1/20 0.40
CLK4 Q9HAZ1 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
ALOX5 P09917 1/20 0.39
OR51E2 Q9H255 1/20 0.39
ADRB2 P07550 1/20 0.39
ADRB1 P08588 1/20 0.39
CYP4F2 P78329 1/20 0.38
CYP4A11 Q02928 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5564662 0.87 TSHR (0.44) PYGLTSHRPTPN1KMT2ACYP11B1
SCHEMBL9558295 0.85 KMT2A (0.51) PYGLTSHRKMT2ASIRT2CDK8
SCHEMBL5522734 0.84 ALDH1A1 (0.50) TSHRKMT2AMAPTL3MBTL1CYP4F2
SCHEMBL3066819 0.84 TSHR (0.58) PYGLTSHRPTPN1CYP11B1CYP11B2
SCHEMBL1745477 0.81 CA2 (0.52) ALOX5OR51E2
SCHEMBL14461366 0.81 RAB9A (0.48) PYGLTSHRPTPN1CYP11B1CYP11B2
SCHEMBL23665899 0.80 CYP3A4 (0.49) PYGLTSHRPTPN1KMT2ACYP11B1
SCHEMBL26641492 0.80 CDK8 (0.52) KMT2AMAPTCDK8CLK4ALOX5
SCHEMBL30643734 0.80 CDK8 (0.52) KMT2AMAPTCDK8CLK4ALOX5
SCHEMBL24133079 0.80 L3MBTL1 (0.41) PYGLTSHRKMT2ACYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5260277-A Cell receptor antagonists TANABE SEIYAKU CO., LTD. (JP) 1993-11-09 US disclosed
WO-1993008823-A1 GUANIDINYL AND RELATED CELL ADHESION MODULATION COMPOUNDS TANABE SEIYAKU CO., LTD. (JP) 1993-05-13 WO disclosed