SCHEMBL9548079

SCHEMBL9548079

CSc1cc(C(O)CNC(C)CCc2ccccc2)ccc1C

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 8/20 0.57
ADRA1A P35348 6/20 0.57
ADRB1 P08588 4/20 0.57
ADRA1D P25100 4/20 0.57
ADRA1B P35368 4/20 0.57
ALDH1A1 P00352 3/20 0.57
CYP2D6 P10635 3/20 0.57
ADRA2A P08913 3/20 0.57
LMNA P02545 3/20 0.57
HTR1A P08908 3/20 0.57
SLC6A2 P23975 3/20 0.57
KDM4E B2RXH2 2/20 0.57
HPGD P15428 2/20 0.57
HSD17B10 Q99714 2/20 0.57
OPRM1 P35372 2/20 0.57
DRD3 P35462 2/20 0.57
HTR2B P41595 2/20 0.57
SLC6A3 Q01959 2/20 0.57
CYP1A2 P05177 2/20 0.57
NFKB1 P19838 2/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10648836 0.88 ADRB2 (0.66) ADRB2ADRA1AADRB1ADRA1DADRA1B
SCHEMBL9548053 0.87 SLC6A4 (0.60) ADRB2ADRA1AADRB1CYP2D6HTR1A
Acetic Acid SCHEMBL10652049 0.84 ADRB2 (0.67) ADRB2ADRA1AADRB1ADRA1DADRA1B
SCHEMBL11470324 0.81 ADRB2 (0.59) ADRB2ADRA1AADRB1ADRA1DADRA1B
SCHEMBL8985958 0.80 ADRB1 (0.80) ADRB2ADRA1AADRB1ADRA1DADRA1B
Hydrochloric Acid SCHEMBL11480657 0.78 ADRB2 (0.68) ADRB2ADRA1AADRB1ADRA1DADRA1B
Hydrochloric Acid SCHEMBL11480654 0.78 ADRB2 (0.68) ADRB2ADRA1AADRB1ADRA1DADRA1B
Hydrochloric Acid SCHEMBL11480322 0.78 ADRA1A (0.63) ADRB2ADRA1AADRB1ADRA1DADRA1B
SCHEMBL11470328 0.77 ADRB2 (0.60) ADRB2ADRA1AADRB1ADRA1DADRA1B
SCHEMBL11020328 0.77 ADRB2 (0.63) ADRB2ADRA1AADRB1ADRA1DADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5198587-A Adrenergic Blocking Agents, Hypotensive Agents YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1993-03-30 US disclosed
US-5063246-A Hypotensive YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1991-11-05 US disclosed
US-4880841-A ADRENERGIC BLOCKING AGENTS, HYPOTENSIVE AGENTS YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1989-11-14 US disclosed