SCHEMBL9549922

SCHEMBL9549922

COc1cc(Br)c2c(c1)C1CCN(C)C(C1)N2C

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.33
MMP1 P03956 1/20 0.31
MMP9 P14780 1/20 0.31
MMP13 P45452 1/20 0.31
ADAM17 P78536 1/20 0.31
DRD2 P14416 2/20 0.31
GRM2 Q14416 1/20 0.31
HTR2C P28335 1/20 0.30
MAOA P21397 1/20 0.30
MAOB P27338 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9549895 0.86 SIGMAR1 (0.35) SIGMAR1DRD2HTR2C
SCHEMBL9550063 0.85 SIGMAR1 (0.32) SIGMAR1DRD2HTR2C
SCHEMBL9549952 0.85 ACHE (0.35) MMP1MMP9MMP13ADAM17
SCHEMBL9549981 0.82 SIGMAR1 (0.31) SIGMAR1
SCHEMBL9549983 0.80 ALDH1A1 (0.38) MAPT
SCHEMBL9550005 0.80 FDFT1 (0.37) SIGMAR1DRD2
Acetic Acid SCHEMBL9549945 0.77
SCHEMBL10591290 0.69 ACHE (0.32) SIGMAR1
SCHEMBL9549940 0.67 ACHE (0.42)
SCHEMBL9549885 0.67

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5264575-A Reacting 1,3-benzodiazocine-8-ol derivative with lutidine/2,6-/, triisoproylsilyltrifluoro methane, formed intermediate reacted with lithium chloride, tetrabutylammonium fluoride and isocyanate HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1993-11-23 US disclosed
US-5097033-A Aminoethyl quinoline 2-ones, intermediates for analgesic, and cholinergic agents for memory disorders HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1992-03-17 US disclosed
US-5010083-A Cognition activator; Alzheimer*s disease HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-04-23 US disclosed
EP-0335292-A2 2,6-Methano-1,3-benzodiazocines, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-10-04 EP disclosed