SCHEMBL9549940

SCHEMBL9549940

CC(=O)Oc1ccc2c(c1)C1CCN(C)C(C1)N2C

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ACHE P22303 15/20 0.42
OPRM1 P35372 4/20 0.39
OPRD1 P41143 2/20 0.39
OPRK1 P41145 2/20 0.35
BCHE P06276 4/20 0.35
KDM4E B2RXH2 3/20 0.35
CYP2D6 P10635 2/20 0.35
MEN1 O00255 1/20 0.35
CYP1A2 P05177 1/20 0.35
KMT2A Q03164 1/20 0.35
HIF1A Q16665 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
PTGS1 P23219 1/20 0.35
BLM P54132 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9549952 0.81 ACHE (0.35) ACHEOPRM1OPRD1
SCHEMBL9549900 0.78 KDM4E (0.39) ACHEKDM4ECYP2D6MEN1CYP1A2
SCHEMBL9549934 0.69 BCHE (0.42) ACHEBCHECYP2D6CYP1A2ALDH1A1
SCHEMBL20245487 0.66 ACHE (0.40) ACHEOPRM1OPRD1
SCHEMBL12059730 0.66 ACHE (0.55) ACHEOPRM1OPRK1BCHEKDM4E
SCHEMBL12043451 0.66 ACHE (0.55) ACHEBCHELMNA
SCHEMBL7904755 0.66 ACHE (0.55) ACHEOPRM1OPRK1BCHEKDM4E
Acetic Acid SCHEMBL9549945 0.66
SCHEMBL11162905 0.65 LMNA (0.49) ACHEOPRM1OPRD1OPRK1KDM4E
SCHEMBL9549983 0.64 ALDH1A1 (0.38) KDM4EMEN1CYP1A2KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5010083-A Cognition activator; Alzheimer*s disease HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-04-23 US claimed
US-5264575-A Reacting 1,3-benzodiazocine-8-ol derivative with lutidine/2,6-/, triisoproylsilyltrifluoro methane, formed intermediate reacted with lithium chloride, tetrabutylammonium fluoride and isocyanate HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1993-11-23 US disclosed
US-5097033-A Aminoethyl quinoline 2-ones, intermediates for analgesic, and cholinergic agents for memory disorders HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1992-03-17 US disclosed
US-5010083-A Cognition activator; Alzheimer*s disease HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-04-23 US disclosed
EP-0335292-A2 2,6-Methano-1,3-benzodiazocines, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-10-04 EP disclosed