SCHEMBL9550244

SCHEMBL9550244

COC(=O)/C(=C\N(C)C)N(C)c1nc(-c2ccc(Cl)cc2)c(Br)s1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.38
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 2/20 0.38
PKM P14618 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
NPC1 O15118 3/20 0.36
RAB9A P51151 3/20 0.36
DHODH Q02127 1/20 0.36
PTGDR2 Q9Y5Y4 5/20 0.35
MAPT P10636 1/20 0.34
CYP11B1 P15538 3/20 0.33
CYP11B2 P19099 2/20 0.33
LMNA P02545 2/20 0.33
NPSR1 Q6W5P4 1/20 0.33
GPBAR1 Q8TDU6 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
F2 P00734 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9196621 1.00 SMN1; SMN2 (0.38) SMN1; SMN2KDM4EALDH1A1PKML3MBTL1
SCHEMBL9550208 0.79 NPC1 (0.62) L3MBTL1NPC1RAB9AMAPTMEN1
SCHEMBL9550207 0.79 NPC1 (0.62) L3MBTL1NPC1RAB9AMAPTMEN1
SCHEMBL9362075 0.78 KDM4E (0.42) KDM4EPKMRAB9AMAPTLMNA
SCHEMBL9587765 0.78 KDM4E (0.42) KDM4EPKMRAB9AMAPTLMNA
SCHEMBL10394271 0.78 DHODH (0.45) SMN1; SMN2KDM4EALDH1A1PKML3MBTL1
SCHEMBL10394270 0.78 DHODH (0.45) SMN1; SMN2KDM4EALDH1A1PKML3MBTL1
SCHEMBL9550218 0.74 PTGDR2 (0.40) SMN1; SMN2KDM4EALDH1A1PKML3MBTL1
SCHEMBL9192255 0.73 ALOX15 (0.34) KDM4EALDH1A1L3MBTL1NPC1RAB9A
SCHEMBL9191662 0.73 CNR1 (0.45) SMN1; SMN2L3MBTL1NPC1RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5196541-A PROCESS FOR THE PREPARATION OF SUBSTITUTED 3-AMINOACRYLIC ESTERS BAYER AKTIENGESELLSCHAFT (DE) 1993-03-23 US disclosed