SCHEMBL9555772

SCHEMBL9555772

CC(C)(C)C(=O)OCn1c(C(F)(F)F)nc2ccc(CBr)cc2c1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.39
POLB P06746 1/20 0.39
GAA P10253 1/20 0.39
ALDH1A1 P00352 5/20 0.34
KDM4E B2RXH2 4/20 0.34
HPGD P15428 2/20 0.34
HSD17B10 Q99714 2/20 0.34
CYP2C9 P11712 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C19 P33261 1/20 0.33
NPC1 O15118 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
ACSS2 Q9NR19 1/20 0.33
APEX1 P27695 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC7 Q8WUI4 1/20 0.33
HDAC2 Q92769 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8490703 0.86 SMN1; SMN2 (0.43) NPSR1POLBGAAALDH1A1KDM4E
SCHEMBL9253194 0.76 LMNA (0.43) SMN1; SMN2HDAC3HDAC4HDAC1HDAC7
SCHEMBL9248248 0.75 ALDH1A1 (0.45) NPSR1POLBGAAALDH1A1KDM4E
SCHEMBL9697181 0.75 SMN1; SMN2 (0.43) NPSR1POLBGAAALDH1A1KDM4E
SCHEMBL9245910 0.72 POLB (0.45) NPSR1POLBGAAALDH1A1KDM4E
SCHEMBL9221651 0.71 TYMS (0.43) POLBALDH1A1KDM4EHPGDHSD17B10
SCHEMBL8488725 0.71 MAPT (0.38) POLBGAAALDH1A1KDM4EHPGD
SCHEMBL10431211 0.71 HDAC6 (0.46) NPSR1POLBGAAALDH1A1HPGD
SCHEMBL9515641 0.71 POLB (0.41) NPSR1POLBGAAALDH1A1KDM4E
SCHEMBL8488726 0.71 ALDH1A1 (0.37) GAAALDH1A1KDM4EHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5187167-A Antitumor agents IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-02-16 US disclosed
US-5081124-A Amino acid and polyamino acid derivatives, inhibitors of thymidylate synthetase IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-01-14 US disclosed
EP-0239362-B1 ANTI-TUMOR AGENTS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-12-04 EP disclosed
US-4992550-A Thymidylate synthetase inhibitors IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-02-12 US disclosed
EP-0239362-A2 Anti-tumor agents IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1987-09-30 EP disclosed