SCHEMBL9559459

SCHEMBL9559459

CCOC(=O)CC(CCC(=O)O)NC(=O)Oc1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.52
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
CYP2D6 P10635 2/20 0.41
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
CYP3A4 P08684 1/20 0.41
GAA P10253 1/20 0.41
FAAH O00519 1/20 0.41
ALDH1A1 P00352 2/20 0.40
TSHR P16473 1/20 0.40
SLC1A3 P43003 1/20 0.40
HPGD P15428 2/20 0.39
RAB9A P51151 2/20 0.39
NPC1 O15118 1/20 0.39
CRHBP P24387 1/20 0.39
CRHR2 Q13324 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
POLB P06746 1/20 0.39
MIF P14174 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23129807 0.77 L3MBTL1 (0.57) CYP1A2MEN1KMT2ACYP2D6CYP2C9
SCHEMBL21891791 0.77 L3MBTL1 (0.57) CYP1A2MEN1KMT2ACYP2D6CYP2C9
SCHEMBL5658218 0.75 CYP1A2 (0.59) CYP1A2MEN1KMT2ACYP2D6CYP2C9
SCHEMBL28665914 0.75 CTRB1 (0.56) ALDH1A1MAPK1
SCHEMBL28665913 0.75 CTRB1 (0.56) ALDH1A1MAPK1
SCHEMBL20901379 0.75 CYP1A2 (0.61) CYP1A2MEN1KMT2ACYP2D6CYP2C9
SCHEMBL5113566 0.75 CYP1A2 (0.73) CYP1A2MEN1KMT2ACYP2D6CYP2C9
SCHEMBL22193661 0.73 CTRB1 (0.53) ALDH1A1ALOX15
SCHEMBL9597177 0.73 PLA2G2C (0.41) CYP1A2
SCHEMBL21891842 0.73 CYP1A2 (0.44) CYP1A2MEN1KMT2ACYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0549727-A1 CARBOXYLIC ACID ESTERS OF RAPAMYCIN AMERICAN HOME PRODUCTS CORPORATION (US) 1993-07-07 EP disclosed
US-5130307-A Antibody inhibitors; treating organ graft rejection, fungal infections; antiinflammatory agents AMERICAN HOME PRODUCTS CORPORATION (US) 1992-07-14 US disclosed
WO-1992005179-A1 CARBOXYLIC ACID ESTERS OF RAPAMYCIN AMERICAN HOME PRODUCTS CORPORATION (US) 1992-04-02 WO disclosed