SCHEMBL9562969

SCHEMBL9562969

CCCc1nc2ncc(Br)nc2c(=O)[nH]1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4C Q9H3R0 1/20 0.43
NOS1 P29475 3/20 0.38
MAPK1 P28482 2/20 0.37
HPGD P15428 2/20 0.36
HTT P42858 1/20 0.36
PARP1 P09874 1/20 0.35
GLA P06280 1/20 0.34
PI4KA P42356 1/20 0.34
PI4K2B Q8TCG2 1/20 0.34
PI4K2A Q9BTU6 1/20 0.34
PI4KB Q9UBF8 1/20 0.34
ALDH1A1 P00352 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HSD17B10 Q99714 1/20 0.33
ADORA3 P0DMS8 2/20 0.33
ADORA2A P29274 2/20 0.33
ADORA1 P30542 2/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16333642 0.88 NOS1 (0.40) NOS1HPGDGLAALDH1A1SMN1; SMN2
SCHEMBL3528801 0.73 NOS1 (0.57) NOS1HPGDGLAALDH1A1HSD17B10
SCHEMBL28252089 0.68 XDH (0.56) ALDH1A1
SCHEMBL25903530 0.68 NOS1 (0.47) NOS1HPGDALDH1A1SMN1; SMN2HSD17B10
SCHEMBL1520051 0.68 NOS1 (0.68) NOS1HPGDALDH1A1HSD17B10KMT2A
SCHEMBL24629160 0.67 ALDH1A1 (0.52) NOS1HPGDALDH1A1SMN1; SMN2HSD17B10
SCHEMBL9406903 0.67 PI4KA (0.44) KDM4CNOS1MAPK1PI4KAPI4K2B
SCHEMBL16333912 0.66 ALDH1A1 (0.49) MAPK1HPGDHTTALDH1A1SMN1; SMN2
SCHEMBL9197478 0.66 ALDH1A1 (0.45) NOS1HPGDALDH1A1SMN1; SMN2
SCHEMBL6933543 0.66 KDM4C (0.54) KDM4CHPGDHTTPARP1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0537937-A2 Substituted pyrazino 2,3-D pyrimidinones as angiotensin II antagonists MERCK & CO. INC. (US) 1993-04-21 EP disclosed