SCHEMBL956333

SCHEMBL956333

NC(=O)CCCCc1cccc(-c2nnn[nH]2)c1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PLA2G10 O15496 1/20 0.37
PLA2G2A P14555 1/20 0.37
CES1 P23141 4/20 0.37
NCEH1 Q6PIU2 1/20 0.37
FAAH O00519 3/20 0.36
HDAC6 Q9UBN7 2/20 0.36
PARP1 P09874 1/20 0.36
AURKA O14965 1/20 0.36
SPHK2 Q9NRA0 1/20 0.35
FFAR1 O14842 1/20 0.35
HDAC1 Q13547 3/20 0.35
MAPT P10636 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
DAGLA Q9Y4D2 1/20 0.34
MMP2 P08253 1/20 0.34
MMP9 P14780 1/20 0.34
MMP8 P22894 1/20 0.34
MMP13 P45452 1/20 0.34
MPO P05164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL950000 0.92 FFAR1 (0.39) PLA2G10PLA2G2APARP1AURKAFFAR1
SCHEMBL6957851 0.84 IGF1R (0.39) CES1NCEH1FAAHMMP2MMP9
SCHEMBL6952118 0.82 IGF1R (0.38) CES1NCEH1FAAHMAPTRXFP1
SCHEMBL6954931 0.82 IGF1R (0.38) CES1NCEH1FAAHMAPTRXFP1
SCHEMBL3822509 0.81 SPHK2 (0.31) SPHK2
SCHEMBL949482 0.81 MPO (0.36) FAAHMPO
SCHEMBL6957496 0.80 LPL (0.44) SPHK2
SCHEMBL6952046 0.80 HSD11B1 (0.39) SPHK2
SCHEMBL7379228 0.79 PIM1 (0.38) PARP1
SCHEMBL5438306 0.78 SPHK2 (0.32) SPHK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011006935-A2 TETRAZOLE DERIVATIVES MERCK SERONO S.A. (CH) 2011-01-20 WO disclosed