SCHEMBL9564786

SCHEMBL9564786

CCOC(=O)N1CCC(Nc2nc3ncnc(Cl)c3n2Cc2ccc(F)cc2)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.47
GAA P10253 4/20 0.47
KDM4E B2RXH2 4/20 0.47
MAPT P10636 4/20 0.47
NOS2 P35228 4/20 0.46
NOS1 P29475 3/20 0.46
LMNA P02545 3/20 0.46
MAPK14 Q16539 1/20 0.46
HSD17B10 Q99714 3/20 0.45
HPGD P15428 2/20 0.45
CASP1 P29466 1/20 0.45
CASP7 P55210 1/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
MAP4K4 O95819 1/20 0.45
SMN1; SMN2 Q16637 4/20 0.44
HTT P42858 3/20 0.44
NPSR1 Q6W5P4 1/20 0.44
NOS3 P29474 1/20 0.43
MEN1 O00255 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9564937 0.83 HSD17B10 (0.47) ALDH1A1GAAKDM4EMAPTLMNA
SCHEMBL9698218 0.82 GAA (0.55) ALDH1A1GAAKDM4EMAPTNOS2
SCHEMBL9564865 0.80 SSTR5 (0.63) GAAKDM4EMAPTLMNASMN1; SMN2
SCHEMBL9630400 0.80 GAA (0.53) ALDH1A1GAAKDM4EMAPTNOS2
SCHEMBL9564902 0.79 USP2 (0.51) ALDH1A1GAAKDM4EMAPTNOS2
SCHEMBL6995354 0.79 LMNA (0.71) ALDH1A1GAAKDM4EMAPTLMNA
SCHEMBL11278989 0.78 LMNA (0.55) ALDH1A1GAAKDM4EMAPTNOS2
SCHEMBL11278216 0.78 GAA (0.57) ALDH1A1GAAKDM4EMAPTNOS2
SCHEMBL9629419 0.77 USP2 (0.48) ALDH1A1GAAKDM4EMAPTNOS2
SCHEMBL10428791 0.77 LMNA (0.57) ALDH1A1GAAKDM4EMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5258380-A Antiallergens, antihistamines JANSSEN PHARMACEUTICA N.V. (BE) 1993-11-02 US disclosed
EP-0206415-B1 (4-PIPERIDINYLMETHYL AND -HETERO)PURINES JANSSEN PHARMACEUTICA N.V. (BE) 1993-01-27 EP disclosed
US-5041448-A Antiallergens JANSSEN PHARMACEUTICA N.V. (BE) 1991-08-20 US disclosed
EP-0206415-A2 (4-Piperidinylmethyl and -hetero)purines JANSSEN PHARMACEUTICA N.V. (BE) 1986-12-30 EP disclosed