SCHEMBL9564937

SCHEMBL9564937

CCOC(=O)N1CCC(Cc2nc3ncnc(Cl)c3n2Cc2ccc(F)cc2)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.47
CASP1 P29466 1/20 0.47
CASP7 P55210 1/20 0.47
GRIN2B Q13224 2/20 0.43
GAA P10253 3/20 0.42
SMN1; SMN2 Q16637 3/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
MAPT P10636 3/20 0.39
TSHR P16473 2/20 0.39
OPRD1 P41143 1/20 0.39
ALDH1A1 P00352 5/20 0.38
KDM4E B2RXH2 3/20 0.38
LMNA P02545 2/20 0.38
HPGD P15428 2/20 0.38
HTT P42858 2/20 0.38
TP53 P04637 2/20 0.38
TRPC3 Q13507 1/20 0.38
TRPC7 Q9HCX4 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9564876 0.86 HSD17B10 (0.46) HSD17B10CASP1CASP7GRIN2BGAA
SCHEMBL9564786 0.83 ALDH1A1 (0.47) HSD17B10CASP1CASP7GAASMN1; SMN2
SCHEMBL9564912 0.81 HSD17B10 (0.46) HSD17B10CASP1CASP7GRIN2BGAA
SCHEMBL9564890 0.80 ALDH1A1 (0.46) TSHRALDH1A1
SCHEMBL10550194 0.75 KCNH2 (0.46) HSD17B10CASP1CASP7GAASMN1; SMN2
SCHEMBL10553680 0.75 KCNH2 (0.46) HSD17B10CASP1CASP7GAASMN1; SMN2
SCHEMBL9564828 0.70 HRH1 (0.49) GAASMN1; SMN2MEN1KMT2AMAPT
Bromide SCHEMBL9565007 0.70 KCNH2 (0.42) HSD17B10CASP1CASP7GRIN2BALDH1A1
SCHEMBL3971451 0.69 GAA (0.40) HSD17B10GAASMN1; SMN2TSHRALDH1A1
SCHEMBL9564798 0.68 GAA (0.41) HSD17B10CASP1CASP7GRIN2BGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5258380-A Antiallergens, antihistamines JANSSEN PHARMACEUTICA N.V. (BE) 1993-11-02 US disclosed
EP-0206415-B1 (4-PIPERIDINYLMETHYL AND -HETERO)PURINES JANSSEN PHARMACEUTICA N.V. (BE) 1993-01-27 EP disclosed
US-5041448-A Antiallergens JANSSEN PHARMACEUTICA N.V. (BE) 1991-08-20 US disclosed