SCHEMBL9564854

SCHEMBL9564854

O=C(O)Cc1ccc(-c2cnc[nH]c2=O)cc1CC(=O)O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.44
TSHR P16473 2/20 0.44
CYP3A4 P08684 1/20 0.44
GABRA1 P14867 1/20 0.44
NFKB1 P19838 1/20 0.44
GABRR1 P24046 1/20 0.44
GABRR2 P28476 1/20 0.44
GABRA5 P31644 1/20 0.44
GABRB2 P47870 1/20 0.44
GABRA4 P48169 1/20 0.44
KDM4E B2RXH2 1/20 0.43
MAPT P10636 1/20 0.43
PMP22 Q01453 1/20 0.43
PTGS1 P23219 2/20 0.38
HIF1A Q16665 1/20 0.35
CCNC P24863 1/20 0.34
CDK8 P49336 1/20 0.34
PRMT5 O14744 1/20 0.34
WDR77 Q9BQA1 1/20 0.34
SGK1 O00141 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9564754 0.76 PTGS1 (0.39) PTGS1RXRARXRBGRIN2DGRIN3B
SCHEMBL1227645 0.75 CYP3A4 (0.58) ALDH1A1TSHRCYP3A4GABRA1NFKB1
SCHEMBL12263263 0.73 MKNK1 (0.47) ALDH1A1TSHRKDM4ESGK1CAMKK2
SCHEMBL29678121 0.73 RXRA (0.50) TSHRPTGS1LMNAAKR1B1RXRA
SCHEMBL9564742 0.72 THRA (0.36) KDM4EMAPTPTGS1CCNCCDK8
Bromide SCHEMBL9142238 0.72 QDPR (0.44) CYP3A4
SCHEMBL5156156 0.70 PTGS1 (0.59) TSHRPTGS1LMNAAKR1B1RXRA
SCHEMBL6764983 0.70 CYP3A4 (0.53) ALDH1A1TSHRCYP3A4KDM4EMAPT
SCHEMBL3915545 0.70 IDO1 (0.49) CYP3A4KDM4ELMNA
SCHEMBL9141285 0.67 KMT2A (0.55) KDM4EMAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0544166-A2 Cephalosporinderivatives F. HOFFMANN-LA ROCHE AG (CH) 1993-06-02 EP disclosed