SCHEMBL9564855

SCHEMBL9564855

Cc1ccc(S(=O)(=O)N2CCC(Sc3nc4cncnc4n3Cc3ccc(F)cc3)CC2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP2 O75604 13/20 0.49
CYP1A2 P05177 12/20 0.49
CYP3A4 P08684 12/20 0.49
CYP2C9 P11712 10/20 0.49
CYP2C19 P33261 9/20 0.49
LMNA P02545 4/20 0.47
ALOX15 P16050 2/20 0.47
HTT P42858 1/20 0.47
HSD17B10 Q99714 1/20 0.47
MAPK1 P28482 8/20 0.44
ALDH1A1 P00352 4/20 0.44
SMN1; SMN2 Q16637 4/20 0.44
TSHR P16473 3/20 0.44
HIF1A Q16665 2/20 0.44
TP53 P04637 1/20 0.44
HPGD P15428 1/20 0.42
CYP2D6 P10635 2/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.41
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9564962 0.84 USP2 (0.50) USP2CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL9535858 0.83 PKM (0.51) USP2LMNAALOX15HTTHSD17B10
SCHEMBL9565025 0.78 CYP1A2 (0.53) USP2CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL9564873 0.72 CYP1A2 (0.65) USP2CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL9564945 0.71 CYP3A4 (0.54) USP2CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL10795380 0.71 PKM (0.56) LMNAHTTALDH1A1SMN1; SMN2TP53
SCHEMBL8565877 0.69 HSD11B1 (0.46) USP2LMNAMAPK1ALDH1A1SMN1; SMN2
SCHEMBL22039143 0.69 CYP1A2 (0.73) USP2CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL9540017 0.68 PKM (0.54) USP2LMNAALOX15HTTHSD17B10
SCHEMBL2607566 0.67 CYP1A2 (0.49) USP2CYP1A2CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5258380-A Antiallergens, antihistamines JANSSEN PHARMACEUTICA N.V. (BE) 1993-11-02 US disclosed
EP-0206415-B1 (4-PIPERIDINYLMETHYL AND -HETERO)PURINES JANSSEN PHARMACEUTICA N.V. (BE) 1993-01-27 EP disclosed
US-5041448-A Antiallergens JANSSEN PHARMACEUTICA N.V. (BE) 1991-08-20 US disclosed
EP-0206415-A2 (4-Piperidinylmethyl and -hetero)purines JANSSEN PHARMACEUTICA N.V. (BE) 1986-12-30 EP disclosed