SCHEMBL9564922

SCHEMBL9564922

COc1ncnc2c1nc(CC1CCNCC1)n2Cc1ccc(F)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.43
HTR6 P50406 5/20 0.41
TLR7 Q9NYK1 1/20 0.40
CYP3A4 P08684 7/20 0.38
CYP2C9 P11712 5/20 0.38
CASP1 P29466 3/20 0.38
CASP7 P55210 3/20 0.38
HIF1A Q16665 2/20 0.38
NR4A2 P43354 1/20 0.38
CYP1A2 P05177 6/20 0.37
CYP2C19 P33261 4/20 0.37
TSHR P16473 3/20 0.37
PIK3CD O00329 1/20 0.37
USP2 O75604 3/20 0.37
ALDH1A1 P00352 3/20 0.37
HSD17B10 Q99714 3/20 0.37
HPGD P15428 1/20 0.37
MAPK1 P28482 1/20 0.37
HTR1A P08908 1/20 0.36
DRD2 P14416 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9564830 0.85 SSTR5 (0.43) KCNH2
Bromide SCHEMBL9564766 0.84 KCNH2 (0.42) KCNH2HTR6TLR7CYP3A4CYP2C9
SCHEMBL9564851 0.80 CYP1A2 (0.54) KCNH2CYP3A4CYP2C9CASP1CASP7
SCHEMBL9601946 0.76 HTR7 (0.44) KCNH2HTR1ADRD2HTR2AHTR7
Oxalic Acid SCHEMBL9564885 0.75 CYP1A2 (0.51) KCNH2CYP3A4CYP2C9CASP1CASP7
Oxalic Acid SCHEMBL9564888 0.75 CYP1A2 (0.51) KCNH2CYP3A4CYP2C9CASP1CASP7
SCHEMBL9535735 0.74 TP53 (0.51) KCNH2NR4A2
SCHEMBL9564783 0.74 CYP3A4 (0.39) KCNH2HTR6TLR7CYP3A4CYP2C9
Hydrochloric Acid SCHEMBL9537452 0.73 TP53 (0.50) KCNH2NR4A2
SCHEMBL9537829 0.73 KCNH2 (0.58) KCNH2NR4A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5258380-A Antiallergens, antihistamines JANSSEN PHARMACEUTICA N.V. (BE) 1993-11-02 US disclosed
US-5041448-A Antiallergens JANSSEN PHARMACEUTICA N.V. (BE) 1991-08-20 US disclosed
EP-0206415-A2 (4-Piperidinylmethyl and -hetero)purines JANSSEN PHARMACEUTICA N.V. (BE) 1986-12-30 EP disclosed