SCHEMBL9564783

SCHEMBL9564783

CN1CCC(Cc2nc3c(O)ncnc3n2Cc2ccc(F)cc2)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.39
ALDH1A1 P00352 4/20 0.39
HSD17B10 Q99714 3/20 0.39
GLA P06280 1/20 0.39
CYP2D6 P10635 3/20 0.38
KCNH2 Q12809 2/20 0.38
CHRM1 P11229 2/20 0.38
HRH1 P35367 2/20 0.38
STAT3 P40763 1/20 0.38
CYP1A2 P05177 3/20 0.38
TSHR P16473 2/20 0.38
RPS6KB1 P23443 2/20 0.37
USP2 O75604 3/20 0.37
CYP2C19 P33261 2/20 0.37
CYP2C9 P11712 1/20 0.37
PDE10A Q9Y233 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37
HTR6 P50406 1/20 0.36
CASP1 P29466 2/20 0.36
CASP7 P55210 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9564863 0.87 NR4A2 (0.48) KCNH2
Bromide SCHEMBL9564766 0.86 KCNH2 (0.42) CYP3A4ALDH1A1HSD17B10CYP2D6KCNH2
SCHEMBL9564878 0.85 HRH1 (0.49) CYP3A4CYP2D6KCNH2CHRM1HRH1
SCHEMBL9564825 0.79 HTR1A (0.50)
SCHEMBL9565008 0.78 DRD2 (0.50) CYP2D6KCNH2CHRM1HRH1TSHR
SCHEMBL9564927 0.78 P2RX7 (0.44) CYP3A4GLACYP2D6KCNH2CHRM1
SCHEMBL9866073 0.77 CCR3 (0.44) ALDH1A1TSHR
SCHEMBL9564912 0.76 HSD17B10 (0.46) CYP3A4ALDH1A1HSD17B10CYP1A2TSHR
SCHEMBL9564964 0.76 ALDH1A1 (0.46) ALDH1A1
SCHEMBL9564876 0.76 HSD17B10 (0.46) ALDH1A1HSD17B10TSHRCASP1CASP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5258380-A Antiallergens, antihistamines JANSSEN PHARMACEUTICA N.V. (BE) 1993-11-02 US disclosed
US-5041448-A Antiallergens JANSSEN PHARMACEUTICA N.V. (BE) 1991-08-20 US disclosed
EP-0206415-A2 (4-Piperidinylmethyl and -hetero)purines JANSSEN PHARMACEUTICA N.V. (BE) 1986-12-30 EP disclosed