SCHEMBL9565010

SCHEMBL9565010

CC1(C)C=Cc2ccc(Br)cc2C1=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA4 P22748 1/20 0.42
CA7 P43166 1/20 0.42
CA9 Q16790 1/20 0.42
S100A4 P26447 2/20 0.39
TGM2 P21980 1/20 0.37
CES1 P23141 1/20 0.37
PTPRC P08575 1/20 0.35
BCL2 P10415 2/20 0.34
MCL1 Q07820 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
MALT1 Q9UDY8 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
HTR2C P28335 1/20 0.33
PBRM1 Q86U86 1/20 0.32
HSP90AA1 P07900 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9588381 0.86 CA2 (0.42) CA1CA2CA4CA7CA9
SCHEMBL4228062 0.73 ALDH1A1 (0.42) CA1CA2CA7CA9S100A4
SCHEMBL19017207 0.73 HTR2C (0.36) NPSR1HTR2C
SCHEMBL9587813 0.70 CES1 (0.33) CES1MAPK1
SCHEMBL18989196 0.69 HTR2C (0.36) CA2CA9NPSR1HTR2C
SCHEMBL22555671 0.69 PTPRC (0.48) CA1CA2CA4CA7CA9
SCHEMBL9587106 0.68 PPOX (0.40) CA1CA2CA4CA7CA9
SCHEMBL4648894 0.66 PTPRC (0.66) CA1CA2CA4CA7CA9
SCHEMBL30412580 0.66 PTPRC (0.66) CA1CA2CA4CA7CA9
SCHEMBL9587884 0.66 CA1 (0.40) CA1CA2CA4CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5272170-A Tetralones with pharmacological activity J. URIACH & CIA., S.A. (ES) 1993-12-21 US disclosed
US-5208246-A Hypotensive, bronchodilator J. URIACH & CIA. (ES) 1993-05-04 US disclosed
EP-0525768-A1 Tetralones with pharmacological activity J. URIACH & CIA. S.A. (ES) 1993-02-03 EP disclosed
EP-0489300-A2 Tetralones with pharmacological activity J. URIACH & CIA. S.A. (ES) 1992-06-10 EP disclosed