SCHEMBL9588381

SCHEMBL9588381

CC1(C)C=Cc2cc(Br)ccc2C1=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.42
CA9 Q16790 2/20 0.42
CA1 P00915 1/20 0.42
CA4 P22748 1/20 0.42
CA7 P43166 1/20 0.42
S100A4 P26447 2/20 0.39
NPSR1 Q6W5P4 1/20 0.36
PTPRC P08575 1/20 0.35
BCL2 P10415 2/20 0.34
MCL1 Q07820 1/20 0.34
TDP2 O95551 1/20 0.34
MALT1 Q9UDY8 1/20 0.33
TGM2 P21980 1/20 0.33
CES1 P23141 1/20 0.33
HTR2C P28335 1/20 0.33
METAP1 P53582 1/20 0.32
HSP90AA1 P07900 1/20 0.31
TLR9 Q9NR96 1/20 0.31
HTR2B P41595 1/20 0.31
SIGMAR1 Q99720 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9565010 0.86 CA1 (0.42) CA2CA9CA1CA4CA7
SCHEMBL9587884 0.79 CA1 (0.40) CA2CA9CA1CA4CA7
SCHEMBL9587106 0.79 PPOX (0.40) CA2CA9CA1CA4CA7
SCHEMBL4228062 0.73 ALDH1A1 (0.42) CA2CA9CA1CA7S100A4
SCHEMBL18989196 0.73 HTR2C (0.36) CA2CA9NPSR1HTR2CCA12
SCHEMBL9587759 0.72 ABCC9 (0.44)
SCHEMBL9587813 0.70 CES1 (0.33) CES1
SCHEMBL19017207 0.69 HTR2C (0.36) NPSR1HTR2C
SCHEMBL1500055 0.69 S100A4 (0.48) CA2CA9CA1CA4CA7
SCHEMBL2525185 0.66 PTPRC (0.52) CA2CA9CA1CA4CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5272170-A Tetralones with pharmacological activity J. URIACH & CIA., S.A. (ES) 1993-12-21 US disclosed
US-5208246-A Hypotensive, bronchodilator J. URIACH & CIA. (ES) 1993-05-04 US disclosed
EP-0489300-A2 Tetralones with pharmacological activity J. URIACH & CIA. S.A. (ES) 1992-06-10 EP disclosed