SCHEMBL9565097

SCHEMBL9565097

CC1(C)C(=O)c2cc(Br)ccc2C2OC21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.41
CYP1A2 P05177 1/20 0.41
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA4 P22748 1/20 0.38
CA7 P43166 1/20 0.38
CA9 Q16790 1/20 0.38
LMNA P02545 1/20 0.36
EDNRB P24530 2/20 0.36
EDNRA P25101 2/20 0.36
S100A4 P26447 1/20 0.35
PTPRC P08575 1/20 0.35
PBRM1 Q86U86 1/20 0.35
TDP1 Q9NUW8 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
MALT1 Q9UDY8 1/20 0.33
TGM2 P21980 1/20 0.33
CES1 P23141 1/20 0.33
BCHE P06276 1/20 0.32
MEN1 O00255 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9565096 0.88 MAPK1 (0.39) MAPK1CYP1A2CA1CA2CA4
SCHEMBL9588113 0.78 IDO1 (0.41) MAPK1CA1CA2CA7CA9
SCHEMBL9702389 0.72 CA1 (0.41) MAPK1CYP1A2CA1CA2CA4
SCHEMBL9588599 0.72 CA1 (0.41) MAPK1CYP1A2CA1CA2CA4
SCHEMBL9588129 0.72 CA1 (0.38) CA1CA2CA7CA9MALT1
SCHEMBL9587011 0.72 HTT (0.38) LMNAS100A4L3MBTL1CES1SMN1; SMN2
SCHEMBL9588923 0.70 CA2 (0.46) CYP1A2CA1CA2CA4CA7
SCHEMBL22797685 0.69 MAPK1 (0.46) MAPK1CYP1A2EDNRBEDNRAS100A4
SCHEMBL9586565 0.69 TDP2 (0.37) MAPK1CYP1A2CA1CA2CA4
SCHEMBL9588527 0.69 TDP2 (0.35) CA1CA2LMNACYP2C19AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5272170-A Tetralones with pharmacological activity J. URIACH & CIA., S.A. (ES) 1993-12-21 US disclosed
US-5208246-A Hypotensive, bronchodilator J. URIACH & CIA. (ES) 1993-05-04 US disclosed
EP-0525768-A1 Tetralones with pharmacological activity J. URIACH & CIA. S.A. (ES) 1993-02-03 EP disclosed
EP-0489300-A2 Tetralones with pharmacological activity J. URIACH & CIA. S.A. (ES) 1992-06-10 EP disclosed