SCHEMBL9565096

SCHEMBL9565096

CC1(C)C(=O)c2ccc(Br)cc2C2OC21

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.39
LMNA P02545 2/20 0.39
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA4 P22748 1/20 0.38
CA7 P43166 1/20 0.38
CA9 Q16790 1/20 0.38
S100A4 P26447 1/20 0.35
PTPRC P08575 1/20 0.35
CYP1A2 P05177 1/20 0.34
ALDH1A1 P00352 4/20 0.34
POLB P06746 3/20 0.34
TSHR P16473 1/20 0.34
TDP2 O95551 1/20 0.34
MALT1 Q9UDY8 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
PGR P06401 2/20 0.32
TP53 P04637 1/20 0.32
MAPT P10636 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9565097 0.88 MAPK1 (0.41) MAPK1LMNACA1CA2CA4
SCHEMBL9587011 0.81 HTT (0.38) LMNAS100A4ALDH1A1PGRTP53
SCHEMBL9588129 0.81 CA1 (0.38) CA1CA2CA7CA9ALDH1A1
SCHEMBL9586565 0.81 TDP2 (0.37) MAPK1LMNACA1CA2CA4
SCHEMBL9588923 0.79 CA2 (0.46) CA1CA2CA4CA7CA9
SCHEMBL9588113 0.78 IDO1 (0.41) MAPK1CA1CA2CA7CA9
SCHEMBL9588527 0.78 TDP2 (0.35) LMNACA1CA2TDP2
SCHEMBL9587825 0.75 ALDH1A1 (0.38) ALDH1A1POLBMAPTL3MBTL1
SCHEMBL9588047 0.72 CA1 (0.41) MAPK1LMNACA1CA2CA4
SCHEMBL9141916 0.68 HTR2A (0.36) MAPK1LMNAIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5272170-A Tetralones with pharmacological activity J. URIACH & CIA., S.A. (ES) 1993-12-21 US disclosed
US-5208246-A Hypotensive, bronchodilator J. URIACH & CIA. (ES) 1993-05-04 US disclosed
EP-0525768-A1 Tetralones with pharmacological activity J. URIACH & CIA. S.A. (ES) 1993-02-03 EP disclosed
EP-0489300-A2 Tetralones with pharmacological activity J. URIACH & CIA. S.A. (ES) 1992-06-10 EP disclosed