SCHEMBL9565788

SCHEMBL9565788

O=C1CCN(C(=O)c2cc(C(F)(F)F)cc(C(F)(F)F)c2)C(C(O)c2ccc(Cl)cc2)C1

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RHOC P08134 10/20 0.48
RHOA P61586 10/20 0.48
MGLL Q99685 2/20 0.39
TACR1 P25103 3/20 0.37
USP2 O75604 2/20 0.35
CYP3A4 P08684 2/20 0.35
HSD17B10 Q99714 1/20 0.35
CYP2C9 P11712 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8926077 1.00 RHOC (0.48) RHOCRHOAMGLLTACR1USP2
SCHEMBL8923836 1.00 RHOC (0.48) RHOCRHOAMGLLTACR1USP2
SCHEMBL8924659 0.90 RHOC (0.40) RHOCRHOATACR1
SCHEMBL8924315 0.84 HSD17B2 (0.36) MGLLTACR1ALDH1A1
SCHEMBL8925754 0.84 HSD17B2 (0.36) MGLLTACR1ALDH1A1
SCHEMBL8925804 0.83 MTNR1B (0.38) TACR1MEN1KMT2A
SCHEMBL8925221 0.83 MTNR1B (0.38) TACR1MEN1KMT2A
SCHEMBL8926452 0.77 P2RX7 (0.41)
SCHEMBL8926123 0.77 P2RX7 (0.41)
SCHEMBL8939874 0.73 TACR1 (0.41) TACR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0532456-A1 1-Acylpiperidine derivatives and their use as substance P antagonists CIBA-GEIGY AG (CH) 1993-03-17 EP disclosed