SCHEMBL9566569

SCHEMBL9566569

COCCOc1ccc(Br)cc1-c1nc(N)nc(N)n1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.44
PIK3CA P42336 2/20 0.43
POLB P06746 1/20 0.43
PIK3CD O00329 1/20 0.43
PIK3CB P42338 1/20 0.43
PIK3CG P48736 1/20 0.43
AGPAT2 O15120 10/20 0.42
DYRK1A Q13627 1/20 0.39
NPC1 O15118 1/20 0.39
TSHR P16473 1/20 0.39
RAB9A P51151 1/20 0.39
RECQL P46063 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9566545 0.83 RECQL (0.56) DHFRPIK3CAPIK3CDPIK3CBPIK3CG
SCHEMBL9566435 0.82 MGAM (0.54) POLBAGPAT2NPC1TSHRRAB9A
SCHEMBL4291022 0.81 AGPAT2 (0.52) AGPAT2
SCHEMBL11612156 0.80 KDM4E (0.50) DHFRPIK3CAPOLBTSHR
SCHEMBL13957870 0.76 KDM4E (0.46) POLB
SCHEMBL29684606 0.76 KDM4E (0.46) POLB
SCHEMBL30030889 0.75 DHFR (0.43) DHFRPOLBNPC1TSHRRAB9A
SCHEMBL29168726 0.75 DHFR (0.43) DHFRPOLBNPC1TSHRRAB9A
SCHEMBL31053304 0.73 FBP1 (0.44) NPC1TSHRRAB9A
SCHEMBL1516692 0.73 FBP1 (0.44) NPC1TSHRRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0563386-A1 ANTICANCER COMPOSITION AND COMPOUND NIPPON SHINYAKU COMPANY, LIMITED (JP) 1993-10-06 EP disclosed