SCHEMBL9566583

SCHEMBL9566583

O=C(Nc1nc(NC(=O)c2ccccc2)nc(-c2ccccc2)n1)c1ccccc1

nearest known ligand 0.70

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 5/20 0.70
ADORA3 P0DMS8 7/20 0.61
ADORA2A P29274 2/20 0.59
F2 P00734 2/20 0.59
F12 P00748 2/20 0.59
L3MBTL1 Q9Y468 1/20 0.59
ABCG2 Q9UNQ0 1/20 0.59
MEN1 O00255 2/20 0.55
KMT2A Q03164 2/20 0.55
ALDH1A1 P00352 1/20 0.53
PTPN1 P18031 1/20 0.52
LMNA P02545 1/20 0.51
POLB P06746 1/20 0.51
MAPK1 P28482 1/20 0.50
KDM4E B2RXH2 1/20 0.50
TP53 P04637 1/20 0.50
HSD17B10 Q99714 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3299661 0.90 ADORA1 (0.70) ADORA1ADORA3ADORA2AF2F12
SCHEMBL3945635 0.89 ADORA1 (0.60) ADORA1ADORA3ADORA2AF2F12
SCHEMBL9566416 0.86 LMNA (0.59) ADORA1ADORA3F2F12MEN1
SCHEMBL2623151 0.86 KCNK9 (0.55) ADORA1ADORA3F2L3MBTL1MEN1
SCHEMBL25970402 0.83 POLB (0.59) ADORA1ADORA3ADORA2AL3MBTL1MEN1
SCHEMBL6498848 0.82 ADORA1 (1.00) ADORA1ADORA3ADORA2AF2F12
SCHEMBL2623093 0.81 L3MBTL1 (0.64) ADORA1ADORA3ADORA2AF2F12
SCHEMBL22580648 0.81 KMT2A (0.67) ADORA1ADORA3ADORA2AMEN1KMT2A
SCHEMBL14523614 0.80 F2 (0.56) ADORA1ADORA3F2F12L3MBTL1
SCHEMBL7244671 0.79 ALDH1A1 (0.51) ADORA1ADORA3ADORA2AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0563386-A1 ANTICANCER COMPOSITION AND COMPOUND NIPPON SHINYAKU COMPANY, LIMITED (JP) 1993-10-06 EP disclosed