SCHEMBL9567480

SCHEMBL9567480

Cc1c(-c2ccccc2)oc2c(C(=O)NCCCC(=O)NOC(C)(C)C)cccc2c1=O

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 6/20 0.57
ADRA1A P35348 6/20 0.57
ADRA1D P25100 5/20 0.57
ADRA1B P35368 5/20 0.57
LMNA P02545 5/20 0.51
ALDH1A1 P00352 4/20 0.51
MAPT P10636 4/20 0.50
SMN1; SMN2 Q16637 2/20 0.49
GAA P10253 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
KDM4E B2RXH2 2/20 0.49
CYP1A2 P05177 1/20 0.49
CHRM2 P08172 1/20 0.49
CYP3A4 P08684 1/20 0.49
ADRA2A P08913 1/20 0.49
ADORA3 P0DMS8 1/20 0.49
CYP2D6 P10635 1/20 0.49
CHRM1 P11229 1/20 0.49
ACHE P22303 1/20 0.49
SLC6A2 P23975 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8877043 0.84 HTR1A (0.60) HTR1AADRA1AADRA1DADRA1BLMNA
SCHEMBL8875669 0.83 HTR1A (0.62) HTR1AADRA1AADRA1DADRA1BLMNA
SCHEMBL7050353 0.83 HTR1A (0.61) HTR1AADRA1AADRA1DADRA1BLMNA
SCHEMBL8875540 0.81 HTR1A (0.59) HTR1AADRA1AADRA1DADRA1BLMNA
SCHEMBL7052213 0.80 HTR1A (0.58) HTR1AADRA1AADRA1DADRA1BLMNA
SCHEMBL11034050 0.80 HTR1A (0.57) HTR1AADRA1AADRA1DADRA1BLMNA
SCHEMBL10988543 0.78 LMNA (0.57) HTR1AADRA1AADRA1DADRA1BLMNA
SCHEMBL10984054 0.78 HTR1A (0.75) HTR1AADRA1AADRA1DADRA1BLMNA
SCHEMBL8876256 0.77 ADRA1A (0.70) HTR1AADRA1AADRA1DADRA1BLMNA
SCHEMBL10991960 0.76 HTR1A (0.72) HTR1AADRA1AADRA1DADRA1BLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993017007-A1 HETEROBICYCLIC COMPOUNDS RECORDATI INDUSTRIA CHIMICA E FARMACEUTICA S.P.A. (IT) 1993-09-02 WO disclosed
EP-0558245-A1 Heterobicyclic compounds as antagogists of alpha-1 adrenergic and SHT1A receptors RECORDATI S.A. CHEMICAL and PHARMACEUTICAL COMPANY (CH) 1993-09-01 EP disclosed