SCHEMBL9570618

SCHEMBL9570618

CCOC(=O)C(C(=O)OCC)C(=O)c1c(F)c(F)c(F)c(F)c1Br

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.35
NPSR1 Q6W5P4 2/20 0.35
HTT P42858 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.34
PKM P14618 1/20 0.34
RAB9A P51151 2/20 0.33
GAA P10253 2/20 0.33
NPC1 O15118 1/20 0.33
MITF O75030 1/20 0.33
RECQL P46063 1/20 0.33
HSD17B10 Q99714 1/20 0.33
MTOR P42345 1/20 0.33
ESR1 P03372 1/20 0.32
ALDH1A1 P00352 3/20 0.31
TRPA1 O75762 1/20 0.31
MMP8 P22894 1/20 0.30
AURKA O14965 1/20 0.30
NTRK1 P04629 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10684699 0.88 SMN1; SMN2 (0.39) TP53NPSR1HTTTDP1SMN1; SMN2
SCHEMBL8102404 0.83 TAS1R3 (0.38) TP53NPSR1HTTTDP1SMN1; SMN2
SCHEMBL8111565 0.80 RAB9A (0.36) TP53NPSR1HTTTDP1SMN1; SMN2
SCHEMBL9501097 0.75 NR1H2 (0.38) TP53NPSR1HTTTDP1SMN1; SMN2
SCHEMBL7506823 0.75 MAPT (0.33) NPSR1HTTTDP1PKMRAB9A
SCHEMBL27407281 0.75 TP53 (0.35) TP53NPSR1HTTTDP1SMN1; SMN2
SCHEMBL9135625 0.74 CES2 (0.30)
SCHEMBL332051 0.74 TP53 (0.37) TP53NPSR1HTTTDP1SMN1; SMN2
SCHEMBL17165495 0.72 SMN1; SMN2 (0.48) TP53NPSR1HTTTDP1SMN1; SMN2
SCHEMBL10351474 0.72 HTT (0.34) NPSR1HTTALDH1A1MMP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0550903-A1 Quinolone- and naphthyridone carboxylic acid derivatives as antibacterial agents BAYER AG (DE) 1993-07-14 EP disclosed
CN-1068115-A 7-iso-dihydro-indole-group-quinolone and-1,4 dihydros-1,8 naphthyridine-4-keto carboxylic acid derivatives BAYER AG (DE) 1993-01-20 CN disclosed
EP-0520240-A1 7-Isoindolinyl-quinolone and naphthyridonecarboxylic acid derivatives BAYER AG (DE) 1992-12-30 EP disclosed