SCHEMBL9575366

SCHEMBL9575366

C=C(F)C(=O)Oc1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.44
RXRA P19793 3/20 0.36
RXRB P28702 3/20 0.36
RXRG P48443 3/20 0.36
MAPT P10636 1/20 0.36
KIF11 P52732 1/20 0.35
GPR35 Q9HC97 2/20 0.35
SOD1 P00441 1/20 0.35
TLR8 Q9NR97 2/20 0.34
SCN9A Q15858 3/20 0.33
XPO1 O14980 2/20 0.33
LMNA P02545 1/20 0.33
P2RX1 P51575 1/20 0.33
NOTUM Q6P988 1/20 0.33
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5004362 0.84 ELANE (0.42) CES2RXRARXRBRXRGMAPT
SCHEMBL9575170 0.83 PRSS1 (0.49) CES2MAPTLMNA
SCHEMBL9575659 0.81 KIF11 (0.54) CES2KIF11
SCHEMBL12758749 0.79 PRSS1 (0.38) CES2MAPTKIF11LMNA
SCHEMBL15453834 0.78 CES2 (0.52) CES2RXRARXRBRXRGMAPT
SCHEMBL9575250 0.77 CES2 (0.36) CES2RXRARXRBRXRGMAPT
SCHEMBL7647561 0.76 CES2 (0.50) CES2RXRARXRBRXRGMAPT
SCHEMBL29064876 0.76 CES2 (0.45) CES2RXRARXRBRXRGMAPT
SCHEMBL15836526 0.75 ELANE (0.39) CES2RXRARXRBRXRGMAPT
SCHEMBL9575148 0.75 CYP4F2 (0.41) CES2MAPTSOD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5266668-A Substituted phenyl α-fluoroacrylates HOECHST AKTIENGESELLSCHAFT (DE) 1993-11-30 US disclosed
EP-0249867-B1 SUBSTITUTED PHENYL ESTERS OF ALPHA-FLUOROACRYLIC ACID HOECHST AKTIENGESELLSCHAFT (DE) 1992-01-02 EP disclosed