SCHEMBL9582136

SCHEMBL9582136

CC(C)(C)c1ccc2c(c1)[C@@H]1O[C@H]1C(C)(C)O2

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.36
IDO1 P14902 2/20 0.34
DRD3 P35462 1/20 0.33
HPGD P15428 2/20 0.33
CNR1 P21554 1/20 0.33
CYP19A1 P11511 1/20 0.33
ABCB1 P08183 4/20 0.32
MAPT P10636 1/20 0.32
CNR2 P34972 1/20 0.31
ALOX15 P16050 1/20 0.31
HSD17B10 Q99714 1/20 0.31
TDP1 Q9NUW8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9581542 1.00 ALDH1A1 (0.36) ALDH1A1IDO1DRD3HPGDCNR1
SCHEMBL9582131 1.00 ALDH1A1 (0.36) ALDH1A1IDO1DRD3HPGDCNR1
SCHEMBL9299207 0.86 CYP1A2 (0.37) IDO1ABCB1CNR2
SCHEMBL7768331 0.86 CYP1A2 (0.37) IDO1ABCB1CNR2
SCHEMBL7874514 0.85 IDO1 (0.33) IDO1ABCB1CNR2
SCHEMBL15257382 0.79 ALDH1A1 (0.36) ALDH1A1DRD3HPGDCNR1CYP19A1
SCHEMBL5868357 0.79 IDO1 (0.40) ALDH1A1IDO1ABCB1MAPT
SCHEMBL6274078 0.79 IDO1 (0.40) ALDH1A1IDO1ABCB1MAPT
SCHEMBL5868353 0.79 IDO1 (0.40) ALDH1A1IDO1ABCB1MAPT
SCHEMBL8947014 0.78 IDO1 (0.36) IDO1ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5210234-A Benzopyran intermediates BEECHAM GROUP P.L.C. (GB) 1993-05-11 US disclosed
EP-0250077-B1 PHARMACOLOGICALLY ACTIVE BENZOPYRANES BEECHAM GROUP PLC (GB) 1992-01-02 EP disclosed
US-5075460-A Hypotensive agents BEECHAM GROUP PLC (GB) 1991-12-24 US disclosed
US-4943582-A Active compounds BEECHAM GROUP P.L.C. (GB) 1990-07-24 US disclosed
EP-0250077-A2 Pharmacologically active benzopyranes BEECHAM GROUP PLC (GB) 1987-12-23 EP disclosed