SCHEMBL9299207

SCHEMBL9299207

CC1(C)Oc2ccc(C(F)(F)F)cc2C2OC21

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
CNR2 P34972 1/20 0.35
TERT O14746 1/20 0.34
KCNA5 P22460 1/20 0.34
CHRNB2 P17787 2/20 0.33
CHRNA4 P43681 2/20 0.33
IDO1 P14902 2/20 0.33
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
PNMT P11086 1/20 0.33
HTR2A P28223 3/20 0.33
HTR2C P28335 3/20 0.33
HTR2B P41595 3/20 0.33
BACE1 P56817 1/20 0.32
CYBB P04839 1/20 0.32
NOX3 Q9HBY0 1/20 0.32
NOX4 Q9NPH5 1/20 0.32
NOX1 Q9Y5S8 1/20 0.32
ABCB1 P08183 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7768331 1.00 CYP1A2 (0.37) CYP1A2CYP2D6CNR2TERTKCNA5
SCHEMBL7874514 0.90 IDO1 (0.33) CNR2IDO1ABCB1
SCHEMBL9753193 0.88 TRPV1 (0.36) CNR2CHRNB2CHRNA4IDO1TRPV1
SCHEMBL9582136 0.86 ALDH1A1 (0.36) CNR2IDO1ABCB1
SCHEMBL9582131 0.86 ALDH1A1 (0.36) CNR2IDO1ABCB1
SCHEMBL9581542 0.86 ALDH1A1 (0.36) CNR2IDO1ABCB1
SCHEMBL8137939 0.79 CYP1A2 (0.36) CYP1A2CYP2D6TERTCHRNB2CHRNA4
SCHEMBL7870442 0.78 KCNE1 (0.36) CYP2D6BACE1TRPV1
SCHEMBL7821557 0.78 SERPINE1 (0.40) KCNA5
SCHEMBL5868357 0.78 IDO1 (0.40) IDO1HTR2CHTR2BABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5296492-A Certain chroman derivatives useful for treating symptoms caused by contraction of smooth muscles, circulatory diseases or epilepsy NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1994-03-22 US disclosed
US-5254557-A Administering for reversible airways obstruction and asthma BEECHAM GROUP P.L.C. (GB) 1993-10-19 US disclosed
CN-1068821-A CHROMAN DERIVATIVES NIPPON KAYAKU KK (JP) 1993-02-10 CN disclosed
EP-0518342-A1 Chroman derivatives Nippon Kayaku Kabushiki Kaisha (JP) 1992-12-16 EP disclosed
EP-0373204-A1 NOVEL COMPOUNDS AND TREATMENT BEECHAM GROUP PLC (GB) 1990-06-20 EP disclosed
WO-1989010925-A1 NOVEL COMPOUNDS AND TREATMENT BEECHAM GROUP PLC (GB) 1989-11-16 WO disclosed