SCHEMBL9589604

SCHEMBL9589604

COC(=O)CC(C)C(=O)c1ccc2c(c1)OC(C)C(=O)N2C

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
F10 P00742 6/20 0.38
ITGB3 P05106 6/20 0.38
ITGA2B P08514 6/20 0.38
F2 P00734 6/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C19 P33261 1/20 0.38
RORC P51449 1/20 0.37
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA5 P31644 1/20 0.35
ALDH1A1 P00352 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
TSHR P16473 1/20 0.34
ATM Q13315 1/20 0.34
ABCC8 Q09428 1/20 0.34
KCNJ11 Q14654 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7350849 0.91 CYP3A4 (0.41) F10F2CYP3A4CYP2C19ALDH1A1
SCHEMBL7348843 0.84 CYP3A4 (0.37) F10ITGB3ITGA2BF2CYP3A4
SCHEMBL7343775 0.79 CYP11B2 (0.40) F10RORCGABRG2GABRB3GABRA5
SCHEMBL9589587 0.78 SLC9A1 (0.43) CYP2C19ALDH1A1TSHR
SCHEMBL9589608 0.76 MEN1 (0.32) F10F2ALDH1A1TSHR
SCHEMBL7350852 0.74 MEN1 (0.32) CYP3A4CYP2C19
SCHEMBL7342699 0.72 USP30 (0.46) ALDH1A1TSHR
SCHEMBL7342609 0.72 ALDH1A1 (0.41) CYP3A4CYP2C19ALDH1A1L3MBTL1TSHR
SCHEMBL7412460 0.72 MAPT (0.35) ALDH1A1
SCHEMBL7341558 0.70 ALDH1A1 (0.44) CYP3A4CYP2C19ALDH1A1L3MBTL1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5221742-A PROCESS FOR THE PREPARATION OF 6-(3,4-DIHYDRO-3-OXO-1,4(2H)-BENZOXAZIN-7-YL)-2,3,4,5-TETRAHYDROPYRIDAZIN-3-ONES ORTHO PHARMACEUTICAL CORPORATION (US) 1993-06-22 US disclosed
WO-1992011256-A1 PROCESS FOR THE PREPARATION OF BENZOXAZINYLTETRAHYDROPYRIDAZINES ORTHO PHARMACEUTICAL CORPORATION (US) 1992-07-09 WO disclosed