SCHEMBL9593285

SCHEMBL9593285

O=C(O)C(C(=O)O)C(=O)c1c(F)c(F)c(F)c(F)c1F

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.36
CES1 P23141 1/20 0.36
GAA P10253 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
HTT P42858 2/20 0.33
PKM P14618 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
TSHR P16473 1/20 0.31
LMNA P02545 1/20 0.31
TP53 P04637 1/20 0.31
MAPK1 P28482 1/20 0.31
FOLH1 Q04609 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9135625 0.84 CES2 (0.30) CES2CES1MEN1KMT2A
SCHEMBL20508995 0.72 CES2 (0.39) CES2CES1GAAHTTPKM
SCHEMBL1344949 0.72 PKM (0.46) CES2CES1GAAMEN1KMT2A
SCHEMBL8925773 0.71 AKR1C3 (0.34) CES2CES1
SCHEMBL10137810 0.70 FFAR1 (0.44) CES2CES1GAAHTTPKM
SCHEMBL661258 0.70 CES2 (0.46) CES2CES1GAAMEN1KMT2A
SCHEMBL8471692 0.69 CES2 (0.40) CES2CES1SMN1; SMN2
SCHEMBL10684699 0.69 SMN1; SMN2 (0.39) GAAHTTPKMSMN1; SMN2LMNA
SCHEMBL336394 0.67 CES2 (0.43) CES2CES1GAAMEN1KMT2A
SCHEMBL203915 0.67 CES2 (0.43) CES2CES1GAAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5210193-A Bactericide AMERICAN CYANAMID COMPANY (US) 1993-05-11 US disclosed
US-4940710-A 7-(substituted)piperazinyl-1-ethyl-6-fluoro-1,4-dihydro-4-oxo-3-quinolinecarboxylic acids AMERICAN CYANAMID COMPANY (US) 1990-07-10 US disclosed
EP-0230053-A2 7-(Substituted)piperazinyl-1-ethyl-6-fluoro-1,4-dihydro-4-oxo-3-quinolinecarboxylic acids AMERICAN CYANAMID COMPANY (US) 1987-07-29 EP disclosed