SCHEMBL9600779

SCHEMBL9600779

NC(=O)c1ccc(Cl)nc1N1CCN(CCCC(c2ccc(F)cc2)c2ccc(F)cc2)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 5/20 0.49
HTR2A P28223 4/20 0.49
ADRA1A P35348 4/20 0.49
HRH1 P35367 4/20 0.49
OPRK1 P41145 4/20 0.49
SLC6A3 Q01959 4/20 0.49
CACNA1F O60840 3/20 0.49
DRD4 P21917 3/20 0.49
DRD5 P21918 3/20 0.49
HRH2 P25021 3/20 0.49
ADRA1D P25100 3/20 0.49
HTR7 P34969 3/20 0.49
ADRA1B P35368 3/20 0.49
OPRM1 P35372 3/20 0.49
HTR6 P50406 3/20 0.49
CACNA1D Q01668 3/20 0.49
CACNA1S Q13698 3/20 0.49
CACNA1C Q13936 3/20 0.49
ADORA3 P0DMS8 3/20 0.49
OPRD1 P41143 3/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9602299 0.90 HTR2A (0.52) DRD3HTR2AADRA1AHRH1OPRK1
Hydrochloric Acid SCHEMBL9602476 0.83 DRD3 (0.51) DRD3HTR2AADRA1AHRH1OPRK1
Hydrochloric Acid SCHEMBL9602576 0.80 GRM2 (0.52) DRD3HTR2AADRA1AHRH1OPRK1
Hydrochloric Acid SCHEMBL9601471 0.79 SIGMAR1 (0.48) DRD3HTR2AADRA1AHRH1OPRK1
Hydrochloric Acid SCHEMBL9601482 0.79 SIGMAR1 (0.48) DRD3HTR2AADRA1AHRH1OPRK1
Hydrochloric Acid SCHEMBL9601527 0.75 DRD3 (0.54) DRD3HTR2AADRA1AHRH1OPRK1
SCHEMBL7794415 0.75 DRD3 (0.53) DRD3HTR2AADRA1AHRH1OPRK1
Hydrochloric Acid SCHEMBL11104288 0.74 MEN1 (0.69) DRD3HTR2AADRA1AHRH1OPRK1
SCHEMBL21354137 0.74 KCNH2 (0.57) DRD3HTR2AADRA1AHRH1OPRK1
Hydrochloric Acid SCHEMBL9602489 0.73 OPRM1 (0.59) DRD3HTR2AADRA1AHRH1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0308476-B1 BISPHENYLALKYLPIPERAZINE DERIVATIVES, A METHOD OF THEIR PREPARATION AND A PHARMACEUTICAL PREPARATION Kabi Pharmacia AB (SE) 1993-02-03 EP disclosed