SCHEMBL9602299

SCHEMBL9602299

Cc1ccc(C(N)=O)c(N2CCN(CCCC(c3ccc(F)cc3)c3ccc(F)cc3)CC2)n1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.52
ADRA1A P35348 4/20 0.52
HRH1 P35367 4/20 0.52
DRD3 P35462 4/20 0.52
OPRK1 P41145 4/20 0.52
SLC6A3 Q01959 4/20 0.52
ADORA3 P0DMS8 3/20 0.52
OPRD1 P41143 3/20 0.52
DRD2 P14416 3/20 0.52
CYP3A4 P08684 2/20 0.52
CYP2D6 P10635 2/20 0.52
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
CYP1A2 P05177 2/20 0.52
CYP2C9 P11712 2/20 0.52
KCNH2 Q12809 2/20 0.52
MLNR O43193 1/20 0.52
NR1I2 O75469 1/20 0.52
USP2 O75604 1/20 0.52
LMNA P02545 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9600779 0.90 DRD3 (0.49) HTR2AADRA1AHRH1DRD3OPRK1
Hydrochloric Acid SCHEMBL9602476 0.83 DRD3 (0.51) HTR2AADRA1AHRH1DRD3OPRK1
Hydrochloric Acid SCHEMBL9601471 0.79 SIGMAR1 (0.48) HTR2AADRA1AHRH1DRD3OPRK1
Hydrochloric Acid SCHEMBL9601482 0.79 SIGMAR1 (0.48) HTR2AADRA1AHRH1DRD3OPRK1
Oxalic Acid SCHEMBL9602525 0.78 DRD3 (0.58) HTR2AADRA1AHRH1DRD3OPRK1
SCHEMBL9601090 0.75 CYP3A4 (0.48) HTR2AADRA1AHRH1DRD3OPRK1
SCHEMBL7794415 0.75 DRD3 (0.53) HTR2AADRA1AHRH1DRD3OPRK1
Hydrochloric Acid SCHEMBL9602632 0.74 MEN1 (0.49) HTR2AADRA1AHRH1DRD3OPRK1
Hydrochloric Acid SCHEMBL11104288 0.74 MEN1 (0.69) HTR2AADRA1AHRH1DRD3OPRK1
SCHEMBL21354137 0.74 KCNH2 (0.57) HTR2AADRA1AHRH1DRD3OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0308476-B1 BISPHENYLALKYLPIPERAZINE DERIVATIVES, A METHOD OF THEIR PREPARATION AND A PHARMACEUTICAL PREPARATION Kabi Pharmacia AB (SE) 1993-02-03 EP disclosed