SCHEMBL9601140

SCHEMBL9601140

CCN(C(=O)c1ccc([N+](=O)[O-])cc1F)[C@](CC)(CCC(=O)O)C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.40
TP53 P04637 1/20 0.40
ALDH1A1 P00352 8/20 0.39
GAA P10253 3/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
THRB P10828 1/20 0.39
CYP1A2 P05177 2/20 0.35
CYP2C9 P11712 1/20 0.35
HPGD P15428 1/20 0.35
CYP2C19 P33261 1/20 0.35
KMT2A Q03164 1/20 0.35
MAPT P10636 3/20 0.34
TDP1 Q9NUW8 2/20 0.34
CYP3A4 P08684 1/20 0.34
ALOX15 P16050 1/20 0.34
POLB P06746 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9556472 0.88 HTT (0.41) HTTTP53ALDH1A1GAAL3MBTL1
SCHEMBL8722805 0.75 L3MBTL1 (0.37) HTTTP53ALDH1A1GAAL3MBTL1
SCHEMBL1781383 0.70 L3MBTL1 (0.65) HTTTP53ALDH1A1GAAL3MBTL1
SCHEMBL6311889 0.68 ALDH1A1 (0.36) TP53ALDH1A1THRBCYP1A2CYP2C9
SCHEMBL6308181 0.68 TPMT (0.34) ALDH1A1L3MBTL1THRBCYP1A2HPGD
SCHEMBL16115685 0.68 L3MBTL1 (0.50) HTTTP53ALDH1A1GAAL3MBTL1
SCHEMBL12709974 0.67 ALDH1A1 (0.48) HTTTP53ALDH1A1GAAL3MBTL1
SCHEMBL10965940 0.67 ALDH1A1 (0.38) HTTALDH1A1THRBCYP1A2HPGD
SCHEMBL77925 0.67 ALDH1A1 (0.64) HTTTP53ALDH1A1GAAKMT2A
SCHEMBL25837924 0.67 ALDH1A1 (0.64) HTTTP53ALDH1A1GAAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5236927-A Reduced toxicity; side effect reduction NATIONAL RESEARCH DEVELOPMENT CORPORATION (GB) 1993-08-17 US disclosed
EP-0204529-B1 ANTI-CANCER QUINAZOLINE DERIVATIVES BTG INTERNATIONAL LIMITED (GB) 1993-03-31 EP disclosed
EP-0204529-A2 Anti-cancer quinazoline derivatives BTG INTERNATIONAL LIMITED (GB) 1986-12-10 EP disclosed