SCHEMBL9601289

SCHEMBL9601289

NC1=CN=CNC1(N)Cc1cccs1

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.35
TSHR P16473 2/20 0.33
MGMT P16455 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.32
ADRA1D P25100 2/20 0.32
HSD17B10 Q99714 1/20 0.32
ADRA2A P08913 2/20 0.32
ADRA2B P18089 2/20 0.32
ADRA2C P18825 2/20 0.32
PNP P00491 2/20 0.31
POLB P06746 1/20 0.30
ADORA3 P0DMS8 1/20 0.30
ADORA2A P29274 1/20 0.30
ADORA2B P29275 1/20 0.30
ADORA1 P30542 1/20 0.30
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9602820 0.73 MGMT (0.34) TSHRMGMTPNP
SCHEMBL9601280 0.68 TAAR1 (0.35) TAAR1TSHRMGMTL3MBTL1ADRA1D
SCHEMBL5944840 0.63 TAAR1 (0.36) TAAR1TSHRMGMTL3MBTL1HSD17B10
SCHEMBL31617182 0.62 TAAR1 (0.35) TAAR1TSHRMGMTL3MBTL1ADRA1D
SCHEMBL2030841 0.60 TAAR1 (0.71) TAAR1TSHRL3MBTL1ADRA2AADRA2B
SCHEMBL4457103 0.59 TAAR1 (0.42) TAAR1TSHRMGMTL3MBTL1ADRA1D
SCHEMBL121154 0.57
SCHEMBL17033075 0.56 HSD11B1 (0.43) TAAR1TSHRHSD17B10ADRA2AADRA2B
SCHEMBL30960368 0.56 GRIN2B (0.44) TAAR1L3MBTL1HSD17B10ADRA2AADRA2B
SCHEMBL559559 0.56 TAAR1 (0.56) TAAR1TSHRL3MBTL1ADRA1DHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0206415-B1 (4-PIPERIDINYLMETHYL AND -HETERO)PURINES JANSSEN PHARMACEUTICA N.V. (BE) 1993-01-27 EP disclosed