SCHEMBL9602349

SCHEMBL9602349

O=CC(c1cccnc1)c1cccc(C(F)(F)F)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.48
KCNA5 P22460 4/20 0.47
KCNH2 Q12809 1/20 0.46
TSHR P16473 2/20 0.44
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.44
PNMT P11086 1/20 0.43
CYP19A1 P11511 1/20 0.42
NPY5R Q15761 1/20 0.41
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
MAPT P10636 2/20 0.41
TDP1 Q9NUW8 2/20 0.41
HTT P42858 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CES2 O00748 1/20 0.40
ACP3 P15309 1/20 0.40
VNN1 O95497 1/20 0.40
PIM1 P11309 1/20 0.40
GAA P10253 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6970288 0.86 ACP3 (0.50) TSHRPNMTCES2ACP3
SCHEMBL7555691 0.85 CES2 (0.46) KIF11PNMTL3MBTL1CES2ACP3
SCHEMBL5185325 0.82 ACP3 (0.54) TSHRKMT2AMEN1PNMTALDH1A1
SCHEMBL3905843 0.79 CES2 (0.44) TSHRPNMTCES2ACP3
SCHEMBL7502772 0.79 PNMT (0.42) KCNA5PNMTALDH1A1L3MBTL1CES2
SCHEMBL17593410 0.78 CES2 (0.47) TSHRKMT2AMEN1PNMTCES2
SCHEMBL10558032 0.78 KIF11 (0.51) KIF11KCNA5KCNH2TSHRKMT2A
SCHEMBL3903975 0.78 CYP11B1 (0.44) TSHRCYP19A1NPY5RKDM4EMAPT
SCHEMBL6501170 0.78 CYP19A1 (0.46) KCNA5KMT2AMEN1CYP19A1KDM4E
SCHEMBL4749525 0.77 CES2 (0.46) TSHRKMT2AMEN1PNMTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0221601-B1 [[[(3-Pyridinyl)methylen]amino]oxy]alkanoic acids and esters JANSSEN PHARMACEUTICA N.V. (BE) 1993-03-10 EP disclosed
US-5180832-A Chemical intermediate for thromboxane A2 inhibitor JANSSEN PHARMACEUTICA N.V. (BE) 1993-01-19 US disclosed
US-4746671-A THROMBOXANE SYNTHETASE INHIBITION JANSSEN PHARMACEUTICA N.V. (BE) 1988-05-24 US disclosed