SCHEMBL9602766

SCHEMBL9602766

O=C(c1ccccc1)c1ccn2ccccc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FNTA P49354 3/20 0.49
FNTB P49356 3/20 0.49
POLB P06746 1/20 0.47
AKR1C3 P42330 1/20 0.47
ALDH1A1 P00352 2/20 0.46
GAA P10253 2/20 0.44
MAPT P10636 1/20 0.44
KMT2A Q03164 2/20 0.44
ATM Q13315 2/20 0.41
TDP1 Q9NUW8 2/20 0.41
HSP90AA1 P07900 1/20 0.41
PKM P14618 1/20 0.41
CCR6 P51684 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
TLR9 Q9NR96 1/20 0.41
HTT P42858 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
SRD5A2 P31213 1/20 0.41
CYP2C8 P10632 1/20 0.41
CYP2C9 P11712 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27516303 0.88 FNTA (0.39) FNTAFNTBPOLBALDH1A1GAA
SCHEMBL6791634 0.86 FNTA (0.38) FNTAFNTBPOLBAKR1C3ALDH1A1
SCHEMBL6440948 0.86 MEN1 (0.44) POLBALDH1A1GAAMAPTKMT2A
SCHEMBL1490768 0.82 ALDH1A1 (0.47) FNTAFNTBALDH1A1MAPTKDM4E
SCHEMBL9231407 0.81 BAZ2B (0.41) FNTAFNTBPOLBALDH1A1GAA
SCHEMBL5369223 0.79 KDM4E (0.36) FNTAFNTBPOLBALDH1A1GAA
SCHEMBL6266511 0.78 ALDH1A1 (0.41) FNTAFNTBPOLBALDH1A1GAA
SCHEMBL9749020 0.77 ALDH1A1 (0.41) FNTAFNTBPOLBALDH1A1GAA
SCHEMBL2631222 0.77 MAPT (0.42) POLBALDH1A1GAAMAPTKMT2A
SCHEMBL19714951 0.76 GAA (0.46) ALDH1A1GAAMAPTHTTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0022762-B1 INDOLIZINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR THERAPEUTICAL USE S.A. SANOFI - LABAZ N.V. (BE) 1981-11-25 EP claimed
EP-0022762-A1 Indolizine derivatives, process for their preparation and their therapeutical use S.A. SANOFI - LABAZ N.V. (BE) 1981-01-21 EP claimed
US-5182291-A Angina pectoris, hypotensive, antiarrhythmia, cerebral vascular insufficiency SANOFI (FR) 1993-01-26 US disclosed
US-5147878-A Hypotensive, antiarrhythmia agents SANOFI (FR) 1992-09-15 US disclosed
US-5039700-A Cardiovascular disorders, antitumor agents SANOFI (FR) 1991-08-13 US disclosed
EP-0235111-B1 INDOLIZINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND COMPOSITIONS CONTAINING THEM SANOFI S.A. (FR) 1991-04-10 EP disclosed
US-4957925-A HYPOTENSIVE AGENTS, ANTIARRHYTHMIA AGENTS, TREATMENT OF ANGINA SANOFI (FR) 1990-09-18 US disclosed
EP-0235111-A1 Indolizine derivatives, process for their preparation and compositions containing them SANOFI S.A. (FR) 1987-09-02 EP disclosed
US-4400387-A USEFUL IN VETERINARY MEDICINE FOR TREATMENT OF PSYCHOLOGICAL DISORDERS S. A. LABAZ-SANOFI N.V. (FR) 1983-08-23 US disclosed
EP-0022762-B1 INDOLIZINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR THERAPEUTICAL USE S.A. SANOFI - LABAZ N.V. (BE) 1981-11-25 EP disclosed
EP-0022762-A1 Indolizine derivatives, process for their preparation and their therapeutical use S.A. SANOFI - LABAZ N.V. (BE) 1981-01-21 EP disclosed