SCHEMBL1490768

SCHEMBL1490768

O=C(O)c1ccn2ccccc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.47
ALOX15 P16050 1/20 0.46
FNTA P49354 3/20 0.45
FNTB P49356 3/20 0.45
NOTUM Q6P988 2/20 0.43
PTGS1 P23219 1/20 0.42
PTGS2 P35354 1/20 0.42
KDM4E B2RXH2 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
MAPT P10636 2/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
MYC P01106 2/20 0.40
NR4A1 P22736 1/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
HMGB1 P09429 1/20 0.40
HPGD P15428 1/20 0.40
CA4 P22748 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25514677 0.87 ALDH1A1 (0.50) ALDH1A1ALOX15FNTAFNTBKDM4E
SCHEMBL27516303 0.85 FNTA (0.39) ALDH1A1ALOX15FNTAFNTBNOTUM
SCHEMBL5369223 0.83 KDM4E (0.36) ALDH1A1ALOX15FNTAFNTBNOTUM
SCHEMBL9602766 0.82 FNTA (0.49) ALDH1A1FNTAFNTBKDM4EMAPT
SCHEMBL2631222 0.82 MAPT (0.42) ALDH1A1KDM4EMAPTNPC1HPGD
SCHEMBL9749020 0.82 ALDH1A1 (0.41) ALDH1A1ALOX15FNTAFNTBNOTUM
SCHEMBL9231407 0.82 BAZ2B (0.41) ALDH1A1FNTAFNTBNOTUMKDM4E
Hydrochloric Acid SCHEMBL16468136 0.80 KDM4E (0.41) ALDH1A1KDM4EMAPTNPC1HPGD
SCHEMBL17912676 0.80 CYP3A4 (0.45) ALDH1A1ALOX15FNTAFNTBKDM4E
SCHEMBL30075082 0.79 ALOX15 (0.34) ALDH1A1ALOX15FNTAFNTBPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 112 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106010508-B A kind of indolizine carboxylic acids pH fluorescence probes and its application 泰山医学院 2018-03-27 CN claimed
CN-106010508-A Indolizine carboxylic acid type pH fluorescent probe and application thereof 泰山医学院 2016-10-12 CN claimed
CN-1763039-A Indolizine carboxyl acid analog compound synthesis method UNIV NANJING NORMAL (CN) 2006-04-26 CN claimed
EP-0986560-B1 PYRROLO 2,1,5-CD]INDOLIZINE DERIVATIVES USEFUL IN THE PREVENTION OR TREATMENT OF ESTROGEN RELATED DISEASES OR SYNDROMES KAROBIO AB (SE) 2004-03-24 EP claimed
JP-2002515909-A 2002-05-28 JP claimed
EP-0988303-A1 PYRROLO 2,1,5-cd]INDOLIZINE DERIVATIVES USEFUL IN THE PREVENTION OR TREATMENT OF ESTROGEN RELATED DISEASES OR SYNDROMES NOVO NORDISK A/S (DK) 2000-03-29 EP claimed
WO-1998055483-A1 PYRROLO[2,1,5-cd]INDOLIZINE DERIVATIVES USEFUL IN THE PREVENTION OR TREATMENT OF ESTROGEN RELATED DISEASES OR SYNDROMES NOVO NORDISK A/S (DK) 1998-12-10 WO claimed
EP-0471609-B1 Benzofuran Derivatives, Benzothiophenes, Indoles or Indolizines, Process for Production and Compositions containing them SANOFI SA (FR) 1996-11-27 EP claimed
EP-0471609-A1 Benzofuran Derivatives, Benzothiophenes, Indoles or Indolizines, Process for Production and Compositions containing them SANOFI (FR) 1992-02-19 EP claimed
US-20250042900-A1 INDOLIZINE COMPOUNDS FOR THE TREATMENT OF MENTAL DISORDERS OR INFLAMMATION TACTOGEN INC (US) 2025-02-06 US disclosed
EP-4499058-A2 INDOLIZINE COMPOUNDS FOR THE TREATMENT OF MENTAL DISORDERS OR INFLAMMATION Tactogen Inc. (US) 2025-02-05 EP disclosed
EP-4482832-A1 5-[7-(3,4-DIHYDRO-1H-ISOQUINOLINE-2-CARBONYL)-1,2,3,4 TETRAHYDROISOQUINOLIN-6-Y L]-1H-PYRROLE-3-CARBOXAMIDE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USES AS PRO-APOPTOTIC AGENTS Les Laboratoires Servier (FR) 2025-01-01 EP disclosed
CN-119053587-A 5- [7- (3, 4-Dihydro-1H-isoquinoline-2-carbonyl) -1,2,3,4 tetrahydroisoquinolin-6-yl ] -1H-pyrrole-3-carboxamide derivatives, pharmaceutical compositions containing same and use thereof as pro-apoptotic agents 法国施维雅药厂 2024-11-29 CN disclosed
US-20240308999-A1 INDOLIZINE COMPOUNDS FOR THE TREATMENT OF MENTAL DISORDERS OR MENTAL ENHANCEMENT TACTOGEN INC (US) 2024-09-19 US disclosed
EP-0289170-B1 AZABICYCLIC COMPOUNDS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM BEECHAM GROUP PLC (GB) 1993-06-23 EP disclosed
CN-1018643-B Process for producing sulfonylurea compound TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1992-10-14 CN disclosed
EP-0471609-A1 Benzofuran Derivatives, Benzothiophenes, Indoles or Indolizines, Process for Production and Compositions containing them SANOFI (FR) 1992-02-19 EP disclosed
US-4882327-A NERVOUS SYSTEM DISORDERS BEECHAM GROUP P.L.C. (GB) 1989-11-21 US disclosed
EP-0289170-A2 Azabicyclic compounds, process for their preparation and pharmaceutical compositions containing them BEECHAM GROUP PLC (GB) 1988-11-02 EP disclosed
CN-87102123-A Sulfonylurea compounds, their preparation and their use as herbicides 1987-10-21 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240308999-A1 INDOLIZINE COMPOUNDS FOR THE TREATMENT OF MENTAL DISORDERS OR MENTAL ENHANCEMENT PNMT, HTR5A, HTR4 ALDH1A1 4486/4885ALOX15 679/4885FNTA 1183/4885
US-20250042900-A1 INDOLIZINE COMPOUNDS FOR THE TREATMENT OF MENTAL DISORDERS OR INFLAMMATION TPH2, TPH1, IDO2 ALDH1A1 2187/4885ALOX15 332/4885FNTA 2495/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.