SCHEMBL9602979

SCHEMBL9602979

CC(CN(C)C)Oc1ccc(-n2nc3c(cc2=O)CSc2ccccc2-3)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 1/20 0.43
TOP1 P11387 1/20 0.38
HRH3 Q9Y5N1 2/20 0.35
CA12 O43570 2/20 0.34
CA1 P00915 2/20 0.34
CA2 P00918 2/20 0.34
CA9 Q16790 2/20 0.34
ALDH1A1 P00352 2/20 0.32
KDR P35968 2/20 0.32
KDM4E B2RXH2 1/20 0.32
LMNA P02545 1/20 0.32
HTT P42858 1/20 0.32
CHRM2 P08172 1/20 0.32
ADRA2A P08913 1/20 0.32
CYP2D6 P10635 1/20 0.32
CHRM1 P11229 1/20 0.32
DRD2 P14416 1/20 0.32
ADRA2B P18089 1/20 0.32
ADRA2C P18825 1/20 0.32
CHRM3 P20309 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9865465 0.89 MCHR1 (0.38) MCHR1TOP1HRH3CA12CA1
SCHEMBL9601577 0.88 MCHR1 (0.37) MCHR1TOP1HRH3CA12CA1
SCHEMBL9602962 0.87 HRH3 (0.36) MCHR1HRH3CA12CA1CA2
SCHEMBL9867408 0.87 ALDH1A1 (0.37) MCHR1TOP1CA12CA1CA2
SCHEMBL9866342 0.87 MCHR1 (0.36) MCHR1TOP1HRH3CA12CA1
SCHEMBL9865898 0.87 CA12 (0.35) HRH3CA12CA1CA2CA9
SCHEMBL9866572 0.86 MMP12 (0.40) MCHR1TOP1HRH3CA12CA1
Iodide SCHEMBL10445020 0.86 ALDH1A1 (0.35) HRH3CA12CA1CA2CA9
SCHEMBL9602271 0.86 MCHR1 (0.39) MCHR1TOP1HRH3ALDH1A1LMNA
SCHEMBL9603115 0.85 MCHR1 (0.48) MCHR1TOP1HRH3ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0351435-B1 FUSED PYRIDAZINE COMPOUNDS AND THEIR MEDICINAL USES Yoshitomi Pharmaceutical Industries, Ltd. (JP) 1993-08-04 EP disclosed
US-5045541-A Immunodeficiency disorders YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1991-09-03 US disclosed
EP-0351435-A1 FUSED PYRIDAZINE COMPOUNDS AND THEIR MEDICINAL USES Yoshitomi Pharmaceutical Industries, Ltd. (JP) 1990-01-24 EP disclosed