SCHEMBL9867408

SCHEMBL9867408

COc1ccc(-n2nc3c(cc2=O)CSc2ccc(OC(C)CN(C)C)cc2-3)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.37
CA12 O43570 4/20 0.36
CA1 P00915 4/20 0.36
CA2 P00918 4/20 0.36
CA9 Q16790 4/20 0.36
MCHR1 Q99705 1/20 0.36
MAPT P10636 4/20 0.35
GAA P10253 3/20 0.35
L3MBTL1 Q9Y468 3/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
POLB P06746 1/20 0.35
APEX1 P27695 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
THRB P10828 1/20 0.35
RECQL P46063 1/20 0.35
NPC1 O15118 1/20 0.35
LMNA P02545 1/20 0.35
OPRK1 P41145 1/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9866342 0.93 MCHR1 (0.36) ALDH1A1CA12CA1CA2CA9
SCHEMBL9866572 0.92 MMP12 (0.40) ALDH1A1CA12CA1CA2CA9
SCHEMBL9865465 0.89 MCHR1 (0.38) CA12CA1CA2CA9MCHR1
SCHEMBL9601577 0.89 MCHR1 (0.37) CA12CA1CA2CA9MCHR1
SCHEMBL9602979 0.87 MCHR1 (0.43) ALDH1A1CA12CA1CA2CA9
SCHEMBL9867683 0.85 ALDH1A1 (0.41) ALDH1A1MCHR1MAPTGAAL3MBTL1
SCHEMBL9866266 0.81 MCHR1 (0.42) ALDH1A1MCHR1MAPTGAAL3MBTL1
SCHEMBL9867236 0.80 MCHR1 (0.44) ALDH1A1MCHR1MAPTGAAL3MBTL1
SCHEMBL9866081 0.80 HRH3 (0.33) CA12CA1CA2CA9MMP12
SCHEMBL9602271 0.79 MCHR1 (0.39) ALDH1A1MCHR1MAPTNPC1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5045541-A Immunodeficiency disorders YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1991-09-03 US disclosed
EP-0351435-A1 FUSED PYRIDAZINE COMPOUNDS AND THEIR MEDICINAL USES Yoshitomi Pharmaceutical Industries, Ltd. (JP) 1990-01-24 EP disclosed