SCHEMBL9609110

SCHEMBL9609110

Cc1nn(-c2cccc(NC(=O)C3CC3c3ccccc3)c2)c(C)c1CC(=O)OC(C)(C)C

nearest known ligand 0.79

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 2/20 0.79
P2RX7 Q99572 6/20 0.43
SMN1; SMN2 Q16637 2/20 0.41
LMNA P02545 2/20 0.41
NAMPT P43490 1/20 0.41
ALDH1A1 P00352 1/20 0.41
GAA P10253 1/20 0.41
HTT P42858 1/20 0.41
DGAT2 Q96PD7 1/20 0.41
TSHR P16473 1/20 0.41
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
DEGS1 O15121 1/20 0.39
ACKR3 P25106 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8510947 0.89 PTGDR2 (1.00) PTGDR2P2RX7SMN1; SMN2LMNANAMPT
SCHEMBL8510948 0.89 PTGDR2 (1.00) PTGDR2P2RX7SMN1; SMN2LMNANAMPT
SCHEMBL9608949 0.76 P2RX7 (0.46) PTGDR2P2RX7TSHR
SCHEMBL8516281 0.75 L3MBTL1 (0.53) PTGDR2P2RX7ALDH1A1GAATSHR
SCHEMBL9609107 0.74 P2RX7 (0.47) PTGDR2P2RX7TSHRNPC1RAB9A
SCHEMBL9882891 0.73 AR (0.48) PTGDR2P2RX7TSHRNPC1RAB9A
SCHEMBL9609041 0.73 F2 (0.47) PTGDR2P2RX7ALDH1A1GAAHTT
SCHEMBL9609102 0.71 PDE4B (0.59) P2RX7SMN1; SMN2ALDH1A1TSHRNPC1
SCHEMBL11255334 0.68 TSHR (0.76) P2RX7TSHRNPC1RAB9A
SCHEMBL8511496 0.67 PTGDR2 (0.63) PTGDR2P2RX7LMNAALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069175-A1 NEW PYRAZOLE DERIVATIVES HAVING CRTH2 ANTAGONISTIC BEHAVIOUR ALMIRALL, S.A. (ES) 2012-05-31 WO disclosed
EP-2457900-A1 New pyrazole derivatives having CRTh2 antagonistic behaviour Almirall, S.A. (ES) 2012-05-30 EP disclosed